Phenoxy compounds
Medchemexpress LLC Epertinib hydrochloride | 2071195-74-7 | 98.2% | 596.48 g/mol | C30H28Cl2FN5O3 | 25 MG
Epertinib hydrochloride is a research-grade, orally active, reversible tyrosine kinase inhibitor selective for EGFR, HER2, and HER4. Supplied as a solid hydrochloride salt, it is intended for in vitro and preclinical research and should be handled according to its safety data sheet.
Medchemexpress LLC Epertinib hydrochloride | 2071195-74-7 | 98.2% | 596.48 g/mol | C30H28Cl2FN5O3 | 100 MG
Epertinib hydrochloride is the hydrochloride salt of epertinib, a potent, orally active, reversible, and selective inhibitor of EGFR, HER2, and HER4. It is provided for preclinical research to evaluate signaling pathways and antitumor efficacy and is compatible with click-chemistry applications because of an alkyne functional group.
- Potent, selective tyrosine kinase inhibitor of EGFR, HER2, and HER4.
- Used in preclinical antitumor and signaling research.
- Contains an alkyne moiety compatible with copper-catalyzed azide-alkyne cycloaddition (CuAAC).
- Supplied as a light yellow to yellow solid with high purity.
- Stable under recommended storage: 4°C sealed; in solvent -80°C (6 months), -20°C (1 month).
- Molecular weight 596.48 g/mol; molecular formula C30H28Cl2FN5O3.
Medchemexpress LLC Epertinib hydrochloride | 2071195-74-7 | MFCD32215297 | 98.2% | 596.48 g/mol | C30H28Cl2FN5O3 | 50 MG
Epertinib hydrochloride is a potent, orally active, reversible, and selective tyrosine kinase inhibitor of EGFR, HER2, and HER4 with low-nanomolar IC50 values and demonstrated antitumor activity in preclinical models. The hydrochloride salt is supplied as a solid research compound suitable for biochemical and cell-based studies and contains an alkyne moiety for click chemistry applications.
- Potent inhibition of EGFR, HER2, and HER4 at low-nanomolar concentrations.
- Demonstrated antitumor activity in preclinical in vivo models.
- Contains an alkyne functional group for click chemistry conjugation.
- Supplied as a solid research reagent with high purity.
- Recommended sealed storage away from moisture to preserve stability.
Medchemexpress LLC HY-107367A 10mg Medchemexpress, Epertinib (hydrochloride) CAS:2071195-74-7 Purity:>98%
Medchemexpress, HY-107367A 10mg Epertinib (HCl) CAS:2071195-74-7 Epertinib hydrochloride is a potent, orally active, reversible, and selective tyrosine kinase inhibitor of EGFR, HER2 and HER4, with IC50s of 1.48 nM, 7.15 nM and 2.49 nM, respectively. Epertinib shows potent antitumor activity. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.