Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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511
Tocris Bioscience™ VU 0463271
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and selective KCC2 inhibitor
| Target | KCC2 Inhibitors |
|---|---|
| CAS | 1391737-01-1 |
| Purity | >98% |
| Chemical Name or Material | N-Cyclopropyl-N-(4-methyl-2-thiazolyl)-2-[(6-phenyl-3-pyridazinyl)thio]acetamide |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C19H18N4OS2 |
| Formula Weight | 382.5 |
512
Tocris Bioscience™ GRI 977143
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 325850-81-5 Molecular Formula: C22H17NO4S
| CAS | 325850-81-5 |
|---|---|
| Molecular Formula | C22H17NO4S |
513
Tocris Bioscience™ 2-Hydroxysaclofen
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CAS: 117354-64-0 Molecular Formula: C9H12ClNO4S
| CAS | 117354-64-0 |
|---|---|
| Molecular Formula | C9H12ClNO4S |
514
Tocris Bioscience™ AZD 2461
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CAS: 1174043-16-3 Molecular Formula: C22H22FN3O3
| CAS | 1174043-16-3 |
|---|---|
| Molecular Formula | C22H22FN3O3 |
515
Tocris Bioscience™ CP 376395 hydrochloride
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Potent and selective CRF1 antagonist; binds at an allosteric site
| Inhibitors | CP 376395 hydrochloride |
|---|---|
| Product Type | CP 376395 hydrochloride |
| Molecular Weight (g/mol) | 362.94 |
| Purity | >99% |
516
Tocris Bioscience™ PF 5274857 hydrochloride
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High affinity and selective Smoothened (Smo) receptor antagonist
| Inhibitors | PF 5274857 hydrochloride |
|---|---|
| Product Type | PF 5274857 hydrochloride |
| Molecular Weight (g/mol) | 473.42 |
| Purity | >98% |
517
Tocris Bioscience™ 4-CMTB
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 300851-67-6 Molecular Formula: C14H15ClN2OS
| CAS | 300851-67-6 |
|---|---|
| Molecular Formula | C14H15ClN2OS |
518
Tocris Bioscience™ PK-THPP
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent K2P9.1 (TASK-3) channel blocker
| Product Type | PK-THPP |
|---|---|
| Molecular Weight (g/mol) | 468.59 |
| Purity | >99% |
519
Tocris Bioscience™ TGN 020
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Aquaporin 4 (AQP4) channel blocker
| Inhibitors | TGN 020 |
|---|---|
| Product Type | TGN 020 |
| Molecular Weight (g/mol) | 206.22 |
| Purity | >99% |
520
Tocris Bioscience™ TCH-165
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Enhancer of 20S proteasome assembly and 20S-mediated protein degradation
| Target | Proteasome Modulators |
|---|---|
| CAS | 1446350-60-2 |
| Purity | 0.98 |
| Chemical Name or Material | Ethyl (4 R,5 R)-rel-1-benzyl-5-(4-(benzylamino)phenyl)-2-(4-methoxyphenyl)-4-phenyl-4,5-dihydro-1 H-imidazole-4-carboxylate |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C39H37N3O3 |
521
Tocris Bioscience™ Ebselen
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Glutathione peroxidase mimic; peroxynitrite scavenger
| Inhibitors | Ebselen |
|---|---|
| CAS | 60940-34-3 |
| Product Type | Ebselen |
| Molecular Weight (g/mol) | M.W. (Observed): 274.18 |
| Purity | 98% |
| Recommended Storage | -20°C |
| Molecular Formula | 2-Phenyl-1,2-benzisoselenazol-3(2 H)-one |
522
Tocris Bioscience™ Ibrutinib
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and selective BTK inhibitor (IC50= 0.5 nM)
| CAS | 936563-96-1 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 1-[(3R)-3-[4-Amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl]-1-piperidinyl]-2-propen-1-one |
| Recommended Storage | Store at -20°C |
| Synonym | Agammaglobulinaemia tyrosine kinase, AGMX1, ATKIMD1, B-cell progenitor kinase, BPK, Bruton agammaglobulinemia tyrosine kinase, Bruton tyrosine kinase, dominant-negative kinase-deficient Brutons tyrosine kinase, tyrosine-protein kinase |
| Molecular Formula | C25H24N6O2 |
| Formula Weight | 440.5 |
523
Tocris Bioscience™ ML 204
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 5465-86-1 Molecular Formula: C15H18N2
| CAS | 5465-86-1 |
|---|---|
| Molecular Formula | C15H18N2 |
524
Tocris Bioscience™ BETP
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 1371569-69-5 Molecular Formula: C20H17F3N2O2S
| CAS | 1371569-69-5 |
|---|---|
| Molecular Formula | C20H17F3N2O2S |
525
Tocris Bioscience™ Dexmedetomidine hydrochloride
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 145108-58-3 Molecular Formula: C13H17ClN2
| CAS | 145108-58-3 |
|---|---|
| Molecular Formula | C13H17ClN2 |