Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ Sialyltransferase Inhibitor, 3Fax-Peracetyl Neu5Ac
The Sialyltransferase Inhibitor, 3Fax-Peracetyl Neu5Ac controls the biological activity of Sialyltransferase.
MilliporeSigma™ Calbiochem™ InSolution™ MIF Antagonist, ISO-1
A cell-permeable isoxazoline compound that displays anti-inflammatory properties
MilliporeSigma™ Calbiochem™ Mifepristone
A cell-permeable synthetic steroid that acts as a potent antagonist of progesterone and glucocorticoid receptors.
MilliporeSigma™ Calbiochem™ Lamellipodial Growth Promoter, C8N6 BPA Polyamine
A cell-permeable, fast acting, branched polyamine. Induces growth of actin-enriched lamellipodia within minutes without the need for serum cofactors .
MilliporeSigma™ Calbiochem™ p38 MAP Kinase Inhibitor IV
The p38 MAP Kinase Inhibitor IV, also referenced under CAS 1638-41-1, controls the biological activity of p38 MAP Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Eya2 Phosphatase Inhibitor, MLS000544460
A cell-permeable furylidenebenzohydrazide compound that acts as an inhibitor of Eya2 ED tyrosine phosphatase (IC50
MilliporeSigma™ Calbiochem™ ISR Inhibitor, ISRIB
The cell-permeable, selective inhibitor of eIF2α/eIF2S1 Ser51 phosphorylation-initiated UPR response (≈25 to 200 nM) upon ER stress induction.
MilliporeSigma™ Calbiochem™ Cathepsin Inhibitor III
The Cathepsin Inhibitor III controls the biological activity of Cathepsin. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
MilliporeSigma™ Calbiochem™ AICA-Riboside, 5'-Phosphate
A 5'-phosphorylated analog of membrane permeable AICA-Riboside that mimics AMP and acts as an activator of AMPK (AMP-activated protein kinase).
MilliporeSigma™ Calbiochem™ TLR1/TLR2 Agonist II, CU-T12-9
A diphenyl substituted imidazole based compound that directly and selectively targets TLR1/2 and induces their dimerization and activates TLR1 and 2 signaling leading to NF-κB and AP-1 activation ( K D = 182 and 478 nM, respectively; EC50
MilliporeSigma™ Calbiochem™ 15-PGDH Inhibitor
The 15-PGDH Inhibitor controls the biological activity of 15-PGDH. This small molecule/inhibitor is primarily used for Membrane applications.
MilliporeSigma™ Calbiochem™ CL-387,785
A cell-permeable and irreversible inhibitor of EGF-receptor (EGFR) kinase activity
MilliporeSigma™ Calbiochem™ NF279
A suramin analog that acts as a highly selective, competitive, and reversible ATP-antagonist of P2X receptor (IC50/KB
MilliporeSigma™ Calbiochem™ InSolution™ Gö 6976
Inhibitor of protein kinase C (PKC; IC50 = 7
MilliporeSigma™ Calbiochem™ Dynamin Inhibitor II, MiTMAB
The Dynamin Inhibitor II, MiTMAB, also referenced under CAS 1119-97-7, controls the biological activity of Dynamin. This small molecule/inhibitor is primarily used for Membrane applications.