Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ CL316243 Hydrate
A very potent agonist highly selective for β3 adrenoceptors (EC50 =
MilliporeSigma™ Calbiochem™ Cinnabarinic acid
A partial, low-potency agonist highly selective for mGlu4 receptors (EC50 > 100μM, no effect on other mGlu subtype rece
MilliporeSigma™ Calbiochem™ Leupeptin, Hemisulfate, Microbial
Leupeptin hemisulfate, CAS 103476-89-7, is a reversible inhibitor of trypsin-like proteases and cysteine proteases.
MilliporeSigma™ Calbiochem™ Nimodipine
An L-type Ca2+ channel blocker.
MilliporeSigma™ Calbiochem™ Guanosine 3',5'-cyclic Monophosphate, N2,2'-O-Dibutyryl-, Sodium Salt
Cell-permeable cGMP analog that preferentially activates protein kinase G.
MilliporeSigma™ Calbiochem™ Akt Inhibitor II
The Akt Inhibitor II controls the biological activity of Akt. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Metastin (45-54)
A decapeptide with C-terminally amidated LRF-motif that acts as a potent and selective agonist of AXOR12 and hOT7T175 (a novel human G-protein-coupled receptors).
MilliporeSigma™ Calbiochem™ CDC42 Inhibitor III, ZCL278
A cell-permeable, non-cytotoxic, aqueous soluble (181μM in PBS, pH 7
MilliporeSigma™ Calbiochem™ Celastrol, Celastrus scandens
A cell-permeable dienone-phenolic triterpene compound that exhibits antioxidant and anti-inflammatory properties.
MilliporeSigma™ Calbiochem™ DPDPE
A potent agonist selective for δ opioid receptor (EC50
MilliporeSigma™ Calbiochem™ WAY-100635 Maleate
A selective 5-HT1A receptor antagonist (pKi
MilliporeSigma™ Calbiochem™ VEGFR Tyrosine Kinase Inhibitor VI, AAL-993
The VEGFR Tyrosine Kinse Inhibitor VI, ALL-993, also referenced under CAS 269390-77-4, controls the biological activity of VEGFR Tyrosine Kinase. This small molecule/inhibitor is primarily used for Cancer applications.
MilliporeSigma™ Calbiochem™ InSolution™ Batimastat
A Marimastat type of peptidyl hydroxamate-based inhibitor that potently inhibits a broad-spectrum of metalloproteinases
MilliporeSigma™ Calbiochem™ InSolution™ TLR4 Inhibitor, TAK-242
A 25 mM (2 mg/221 μL) sterile-filtered solution of TLR4 Inhibitor, TAK-242 in DMSO.