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  8. DQP 1105, Tocris Bioscience™

DQP 1105, Tocris Bioscience™

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Quantity:
10mg
50mg
This item is not returnable. View return policy
380560-89-4
C29H24BrN3O4
558.432
CADIBCWPGCNUBD-WEMUOSSPSA-N
4-5-4-bromophenyl-3-2-hydroxy-6-methyl-4-phenylquinolin-3-yl-4,5-dihydro-1h-pyrazol-1-yl-4-oxobutanoic acid,4-5-4-bromophenyl-3-6-methyl-2-oxo-4-phenyl-1,2-dihydroquinolin-3-yl-4,5-dihydro-1h-pyrazol-1-yl-4-oxobutanoic acid,5-4-bromophenyl-3-1,2-dihydro-6-methyl-2-oxo-4-phenyl-3-quinolinyl-4,5-dihydro-gamma-oxo-1h-pyrazole-1-butanoic acid
44657732
4-[(3E)-5-(4-bromophenyl)-3-(6-methyl-2-oxo-4-phenylquinolin-3-ylidene)pyrazolidin-1-yl]-4-oxobutanoic acid
CC1=CC2=C(C(=C3CC(N(N3)C(=O)CCC(=O)O)C4=CC=C(C=C4)Br)C(=O)N=C2C=C1)C5=CC=CC=C5
This item is not returnable. View return policy
380560-89-4
C29H24BrN3O4
558.432
CADIBCWPGCNUBD-WEMUOSSPSA-N
4-5-4-bromophenyl-3-2-hydroxy-6-methyl-4-phenylquinolin-3-yl-4,5-dihydro-1h-pyrazol-1-yl-4-oxobutanoic acid,4-5-4-bromophenyl-3-6-methyl-2-oxo-4-phenyl-1,2-dihydroquinolin-3-yl-4,5-dihydro-1h-pyrazol-1-yl-4-oxobutanoic acid,5-4-bromophenyl-3-1,2-dihydro-6-methyl-2-oxo-4-phenyl-3-quinolinyl-4,5-dihydro-gamma-oxo-1h-pyrazole-1-butanoic acid
44657732
4-[(3E)-5-(4-bromophenyl)-3-(6-methyl-2-oxo-4-phenylquinolin-3-ylidene)pyrazolidin-1-yl]-4-oxobutanoic acid
CC1=CC2=C(C(=C3CC(N(N3)C(=O)CCC(=O)O)C4=CC=C(C=C4)Br)C(=O)N=C2C=C1)C5=CC=CC=C5

Description

GluN2C/GluN2D-selective NMDA antagonist

Noncompetitive NMDA receptor antagonist; displays over 50-fold selectivity for GluN2D- and GluN2C-containing receptors over GluN2B-, GluK2-, GluA1- and GluN2A-containing receptors (IC50 values are 2.7, 8.5, 121, 153, 198 and 206 μM, respectively). Reduces frequency of channel opening.

Please refer to IUPHAR Guide to Pharmacology for the most recent naming conventions.

Quantity 50mg
Formula Weight 558.42
Percent Purity >97%
Chemical Name or Material DQP 1105

Safety and Handling

Recommended Storage : Store at -20°C