GSK 2193874, Tocris Bioscience
Potent and selective TRPV4 antagonist; orally active
Manufacturer: Tocris Bioscience 5106/5
DescriptionPotent and selective TRPV4 antagonist (IC50 values are 2 and 40 nM for rat and human receptors, respectively); inhibits Ca2+ influx through TRPV4 channels. Prevents and reverses pulmonary edema after myocardial infarction in vivo models. Selective over a panel of ~200 human receptors, channels and enzymes. Orally active.
|Observed MW: 691.62|
Safety and Handling
Recommended Storage : Store at 4°C
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