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Tocris™ GSK 5959

Potent and selective BRPF1 inhibitor

Manufacturer:  Tocris™ 5385/10

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Catalog No. 53-851-0

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For Research Use Only



Potent and selective BRPF1 bromodomain inhibitor (IC50 = 80nM). Exhibits >100-fold selectivity for BRPF1 over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains. Inhibits BRPF1 interaction with histone H3.3. Cell permeable.
  • Chemical Name: N-[2,3-Dihydro-1,3-dimethyl-2-oxo-6-(1-piperidinyl)-1H-benzimidazol-5-yl]-2-methoxybenzamide
  • Formula: C22H26N4O3
  • CAS Number: 901245-65-6
  • Solubility: Soluble to 10mM in DMSO with sonication
  • Purity: >99
Description & Specifications


GSK 5959
GSK 5959
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