Tocris™ GSK 5959

Potent and selective BRPF1 inhibitor

Manufacturer: Tocris™ 5385/10

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Catalog No. 53-851-0

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For Research Use Only


    Specifications

    Product Type GSK 5959
    Inhibitors GSK 5959
    Purity >99
    Molecular Weight 394.47
    Quantity 10mg

    Potent and selective BRPF1 bromodomain inhibitor (IC50 = 80nM). Exhibits >100-fold selectivity for BRPF1 over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains. Inhibits BRPF1 interaction with histone H3.3. Cell permeable.

    • Chemical Name: N-[2,3-Dihydro-1,3-dimethyl-2-oxo-6-(1-piperidinyl)-1H-benzimidazol-5-yl]-2-methoxybenzamide
    • Formula: C22H26N4O3
    • CAS Number: 901245-65-6
    • Solubility: Soluble to 10mM in DMSO with sonication
    • Purity: >99

  • Description & Specifications

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