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Tocris Bioscience™ ML 221
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Catalog No. 474810
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47-481-0 10 mg
47-485-0 50 mg
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Catalog No. 47-481-0 Supplier Tocris Bioscience™ Supplier No. 4748/10
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Description

Apelin antagonist

Apelin receptor (APJ) antagonist (IC50 values are 0.70 and 1.75 μM in a cAMP assay and β-arrestin assay, respectively). Displays >37-fold selectivity over the closely related angiotensin II type 1 (AT1) receptor. Exhibits no toxicity towards human hepatocytes at concentrations >50 μM.

Chemical Identifiers

CAS 877636-42-5
Molecular Formula C17H11N3O6S

Specifications

Quantity 10 mg
Formula Weight 385.35
Purity >99%
Molecular Weight (g/mol) 385.35
Chemical Name or Material ML 221

Safety and Handling

Recommended Storage Store at +4°C
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