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  5. Tocris Bioscience™ NVS PAK1 1

Tocris Bioscience™ NVS PAK1 1
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Catalog No. p-7116102
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25 mg
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Catalog No. Quantity
61-322-5 25 mg
61-325 5 mg
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Catalog No. 61-322-5 Supplier Tocris Bioscience™ Supplier No. 6132/25
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Description

Potent and selective PAK1 inhibitor

NVS PAK1 1 is a potent and selective PAK1 inhibitor (IC50 = 5 nM) that displays selective for PAK1 over PAK2 and a panel of 442 kinases. NVS PAK1 1 inhibits autophosphorylation of PAK1 in KRAS-mutated pancreatic cancer cell lines.

A negative control for NVS PAK1 1 is also available; NVS PAK1 C .

Specifications

Chemical Name or Material (3S)-3-(2-Chloro-5-(2,2-difluoroethyl)-8-fluoro-5H-dibenzo[b,e][1,4]diazepin-11-ylamino)-N-isopropylpyrrolidine-1-carboxamide
CAS 1783816-74-9
Assay Percent Range >98%
Quantity 25 mg
Molecular Formula C23H25ClF3N5O
Formula Weight Observed MW: 479.93
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