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Tocris Bioscience™ Penitrem A
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Catalog No. 46171
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Quantity:
1 mg
This item is not returnable. View return policy
This item is not returnable. View return policy

Description

Potent and selective BKCa (KCa1.1) channel blocker

Potent and selective blocker of BKCa (KCa1.1) channels (IC50 values are 6.4 and 64.4 nM for BKCa channels containing α subunits only, and those containing α and β1 respectively). Displays no effect on native delayed rectifier K+ and KATP currents, or cloned KV1.5 channels. Blocks BKCa channels in both inside-out and cell-attached patches. Shown to enhance smooth muscle contraction in vitro and increase total peripheral resistance in vivo.

Chemical Identifiers

CAS 12627-35-9
Molecular Formula C37H44ClNO6

Specifications

Quantity 1 mg
Formula Weight 634.2
Purity >98%
Molecular Weight (g/mol) 634.21
Chemical Name or Material Penitrem A

Safety and Handling

Recommended Storage Store at -20°C
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