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Tocris Bioscience™ Penitrem A

Catalog No. 46171
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46-171 1 mg
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Catalog No. 46-171 Supplier Tocris Bioscience™ Supplier No. 4617/1
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Description

Potent and selective BKCa (KCa1.1) channel blocker

Potent and selective blocker of BKCa (KCa1.1) channels (IC50 values are 6.4 and 64.4 nM for BKCa channels containing α subunits only, and those containing α and β1 respectively). Displays no effect on native delayed rectifier K+ and KATP currents, or cloned KV1.5 channels. Blocks BKCa channels in both inside-out and cell-attached patches. Shown to enhance smooth muscle contraction in vitro and increase total peripheral resistance in vivo.

Chemical Identifiers

CAS 12627-35-9
Molecular Formula C37H44ClNO6

Specifications

Quantity 1 mg
Formula Weight 634.2
Purity >98%
Molecular Weight (g/mol) 634.21
Chemical Name or Material Penitrem A

Safety and Handling

Recommended Storage Store at -20°C
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