Promotional price valid on web orders only. Your contract pricing may differ. Interested in signing up for a dedicated account number?
Learn More
  1. Home
  2. Products
  3. Protein Analysis Reagents
  4. Bioactive Small Molecules
  5. Tocris Bioscience™ PF 915275

Tocris Bioscience™ PF 915275
GREENER_CHOICE

Catalog No. 329110
Change view
Click to view available options
Quantity:
10 mg
50 mg
2 product options available for selection
Product selection table with 2 available options. Use arrow keys to navigate and Enter or Space to select.
Catalog No. Quantity
32-911-0 10 mg
32-915-0 50 mg
Use arrow keys to navigate between rows. Press Enter or Space to select a product option. 2 options available.
2 options
This item is not returnable. View return policy
Catalog No. 32-911-0 Supplier Tocris Bioscience™ Supplier No. 3291/10
Only null left
Add to Cart
Add to Cart
This item is not returnable. View return policy

Description

Potent and selective 11β-hydroxysteroid dehydrogenase inhibitor

Potent and selective 11β-hydroxysteroid dehydrogenase type 1 (11βHSD1) inhibitor (Ki = 2.3 nM) that displays little activity at 11βHSD2 (1.5% inhibition at 10 μM). Inhibits the conversion of prednisone to prednisolone in human hepatocytes in vitro (EC50 = 15 nM) and has antidiabetic activity in vivo. Orally active.

Chemical Identifiers

CAS 857290-04-1
Molecular Formula C18H14N4O2S

Specifications

Quantity 10 mg
Formula Weight 350.39
Purity >98%
Molecular Weight (g/mol) 350.396
Chemical Name or Material PF 915275

Safety and Handling

Recommended Storage Store at Room Temperature
Product Title
Select an issue

By clicking Submit, you acknowledge that you may be contacted by Fisher Scientific in regards to the feedback you have provided in this form. We will not share your information for any other purposes. All contact information provided shall also be maintained in accordance with our Privacy Policy.