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Tocris Bioscience™ PF CBP1

Selective CBP/p300 bromodomain inhibitor

$246.00 - $1035.00

Specifications

Chemical Name or Material 5-(Dimethyl-1,2-oxazol-4-yl)-1-[2-(morpholin-4-yl)ethyl]-2-[2-(4-propoxyphenyl)ethyl]-1H-1,3-benzodiazole
Molecular Formula C29H36N4O3
CAS 1962928-21-7
Product Type Target: Bromodomain Inhibitors
Formula Weight 488.62
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Products 2
Catalog Number Mfr. No. Quantity Price Quantity & Availability  
Catalog Number Mfr. No. Quantity Price Quantity & Availability  
580110 View Documents Tocris Bioscience™
5801/10
10mg Each for $246.00
Add to cart
 
580150 View Documents Tocris Bioscience™
5801/50
50mg Each for $1,035.00
Add to cart
 
Description

Description

Selective CBP/p300 bromodomain inhibitor (IC50 values are 125 and 363 nM, respectively). Exhibits >100-fold selectivity for CBP over BRD4. Also exhibits selectivity over a panel of other bromodomains. Reduces LPS-induced IL-1β, IL-6 and IFN-β expression in macrophages in vitro. Also downregulates RGS4 expression in primary cortical neurons in vitro.

Negative Control also available.

Specifications

Specifications

5-(Dimethyl-1,2-oxazol-4-yl)-1-[2-(morpholin-4-yl)ethyl]-2-[2-(4-propoxyphenyl)ethyl]-1H-1,3-benzodiazole
1962928-21-7
488.62
C29H36N4O3
Target: Bromodomain Inhibitors
Safety and Handling

Safety and Handling

Recommended Storage : Store at 4°C

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