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Tocris Bioscience™ PSB 10 hydrochloride
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Catalog No. 201050
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50 mg
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Catalog No. Quantity
20-105-0 50 mg
20-101-0 10 mg
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Catalog No. 20-105-0 Supplier Tocris Bioscience™ Supplier No. 2010/50
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Description

Potent, highly selective hA3 receptor antagonist/inverse agonist

Potent and highly selective antagonist for the human adenosine A3 receptor, with low affinity for the rat A3 receptor (Ki values are 0.44 and > 17000 nM respectively). Displays > 3800-fold selectivity over human A1, A2A and A2B receptors (Ki values are 4.1, 3.3 and 30 μM respectively) and > 1800-fold selectivity over rat A1 and A2A receptors. Acts as an inverse agonist in the [35S]GTPγS binding assay in hA3-CHO cells (IC50 = 4 nM). Produces thermal hyperalgesia in mice in vivo.

Chemical Identifiers

CAS 591771-91-4
Molecular Formula C16H15Cl4N5O

Specifications

Quantity 50 mg
Formula Weight 435.14
Purity >98%
Molecular Weight (g/mol) 435.13
Chemical Name or Material PSB 10 hydrochloride

Safety and Handling

Recommended Storage Desiccate at +4°C
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