Adenosine receptor inhibitor 1 is a potent and selective adenosine receptor (AR) inhibitor with Ki values of >1000, 68.5, >1000, >1000 nM for A1AR, A2AAR, A2BAR, A3AR, respectively.
- Shows antinociceptive activity.
- Exhibits anti-inflammatory effect.
- Demonstrates peripheral analgesic effect.
- Has potential for the research of cancer or neurodegenerative diseases.