Drug Standards
Selleck Chemical LLC Moxifloxacin (BAY12-8039) HCl S1465-1g
Moxifloxacin (Avelox Avalox BAY12-8039 HCl) is a fourth-generation synthetic fluoroquinolone antibacterial agent
Selleck Chemical LLC Enzalutamide S1250-200mg
Enzalutamide is an androgen-receptor (AR) antagonist with IC50 of 36 nM in LNCaP cells Enzalutamide is shown to increase autophagy
Selleck Chemical LLC Lenalidomide S1029-500mg
Lenalidomide is a TNF- secretion inhibitor with IC50 of 13 nM in PBMCs Lenalidomide (CC-5013) is a ligand of ubiquitin E3 ligase cereblon (CRBN) and it causes selective ubiquitination and degradation of two lymphoid transcription factors IKZF1 and IKZF3 by the CRBN-CRL4 ubiquitin ligase Lenalidomide promotes cleaved caspase-3 expression and inhibit VEGF expression and induces apoptosis
Selleck Chemical LLC Diaveridine S5200-1g
Diaveridine (AI3-23935 CCRIS-3784) is coccidiostat with anti-parasitic activity and also a dihydrofolate reductase (DHFR) inhibitor preventing folic acid synthesis in species of Pneumocystis
Selleck Chemical LLC Fostamatinib (R788) S2625-1g
Fostamatinib (R788) a prodrug of the active metabolite R406 is a Syk inhibitor with IC50 of 41 nM strongly inhibits Syk but not Lyn 5-fold less potent to Flt3 Phase 3
Medchemexpress LLC Tolazamide | 1156-19-0 | 99.9% | 25 MG
Tolazamide is an orally active sulfonylurea agent that inhibits sulfonylurea receptor 1 (SUR1) linked to the inwardly rectifying potassium channel. It has anti-diabetic properties, lowering blood glucose and decreasing insulin dose while maintaining adequate metabolic control. Tolazamide is able to improve or normalize hyperglycemia and HbA.
- Inhibits sulfonylurea receptor 1 (SUR1) linked to the inwardly rectifying potassium channel.
- Possesses anti-diabetic properties.
- Lowers blood glucose.
- Decreases insulin dose while maintaining adequate metabolic control.
- Improves or normalizes hyperglycemia and HbA.
- Attenuates gluconeogenesis and ketogenesis in preclinical studies.
- Soluble in DMSO (≥ 39 mg/mL).
Medchemexpress LLC Vecuronium bromide | 50700-72-6 | 99.9% | 1 ML
Vecuronium bromide is a non-depolarizing neuromuscular blocking agent. It also functions as a nicotinic acetylcholine receptor (nAChR) inhibitor and a muscle relaxant. This compound can be utilized for pre-surgical anesthesia.
- Acts as a nicotinic acetylcholine receptor (nAChR) inhibitor
- Functions as a muscle relaxant
- Can be used for pre-surgical anesthesia
- Inhibits human MATE1-mediated ASP+ uptake
- Inhibits human MATE2K-mediated ASP+ uptake
- Inhibits human OCT2-mediated ASP+ uptake
- Inhibits cancer cell proliferation and migration
Medchemexpress LLC Benzarone | 1477-19-6 | 99.7% | 266.29 | 500 MG
Benzarone is an oral inhibitor of human urate transporter 1 (hURAT1) with an IC50 value of 2.8 μM, and it also functions as an uncoupler of oxidative phosphorylation. This compound has the potential to cause liver damage and can promote cell apoptosis and necrosis. It is utilized to reduce serum uric acid levels and for research related to vascular diseases.
- Oral inhibitor of human urate transporter 1 (hURAT1).
- Functions as an uncoupler of oxidative phosphorylation.
- Used to lower serum uric acid levels.
- Useful for research in vascular diseases.
- May cause liver damage and promote cell apoptosis and necrosis.
Medchemexpress LLC Folic acid | 59-30-3 | 98.4% | 441.40 | 250 MG
Folic acid (Standard) is an analytical standard used as a reference for research and analytical applications. As Vitamin B9, it is an orally active essential nutrient from the B complex group of vitamins. It has shown antidepressant-like effects, and its sodium form can reduce the risk of neonatal neural tube defects. It is also used in research for megaloblastic and macrocytic anemias caused by folic deficiency.
- Analytical standard for assaying
- Used in qualitative, quantitative, and methodological research experiments
- Commonly applied in HPLC, GC, and MS studies
- Essential nutrient from the B complex group (Vitamin B9)
- Shows antidepressant-like effects
- Sodium form reduces the risk of neonatal neural tube defects
- Used in research for megaloblastic and macrocytic anemias
Crescent Chemical Co Inc LIDOCAINE BASE 100 MG
Lignocaine base Pharma./veter. comp. (WS) CAS 137-58-6 Molecular Weight - 234.3373 Storage - RT Catalog Num - DRE-C14629790 chemical
Cayman Chemical ErythromycIn lactobIonate 5g
A macrolide antibiotic and water-soluble form of erythromycin; active against S. aureus and S. pneumoniae, as well as clinical isolates of group A streptococci (MICs = 0.6, 0.06, and 0.031 UG/ml, respectively); increases survival and reduces the number of lung CFUs in a mouse model of S. pneumoniae-induced pneumonia at 50 mg/kg; increases survival in mice infected with P. aeruginosa at 50 or 100 mg/kg
Selleck Chemical LLC Methazolamide 50mg 554-57-4 CL 8490
Methazolamide (CL 8490) is a carbonic anhydrase inhibitor with Ki of 50 nM, 14 nM and 36 nM for hCA I, hCA II and bCA IV isoforms, respectively. *For Research & Development use only. Product is not intended for drug, household, or human consumption.
Crescent Chemical Co Inc DIMETHICONE 1000 250 MG
Dimethicone 1000 Pharma./veter. comp. (WS) CAS 9006-65-9 Molecular Weight - 236.5315 Storage - RT Catalog Num - DRE-C12679100 chemical