Indoles and derivatives
Medchemexpress LLC K-252a | 99533-80-9 | 5 MG
K-252a is a staurosporine analog that inhibits protein kinase with IC50 values of 470 nM for PKC, 140 nM for PKA, 270 nM for Ca2+/calmodulin-dependent kinase type II, and 1.7 nM for phosphorylase kinase. It is also a potent inhibitor (IC50 of 3 nM) of the tyrosine protein kinase (TRK) activity of the NGF receptor gp140trk, which is a product of the trk protooncogene.
- A staurosporine analog.
- Inhibits protein kinase C (PKC) with an IC50 of 470 nM.
- Inhibits protein kinase A (PKA) with an IC50 of 140 nM.
- Inhibits Ca2+/calmodulin-dependent kinase type II with an IC50 of 270 nM.
- Inhibits phosphorylase kinase with an IC50 of 1.7 nM.
- Potent inhibitor of the tyrosine protein kinase (TRK) activity of the NGF receptor gp140trk with an IC50 of 3 nM.
- Appears as a white to light yellow solid.
Sigma Aldrich Fine Chemicals Biosciences K-252a from Nonomuraea longicatena, >=98% (HPLC) | 99533-80-9 | MFCD00161522 | 100UG
K-252a from Nonomuraea longicatena, >=98% (HPLC) | Purity: >=98% (HPLC) | Mol Wt: 467.47 | 99533-80-9 | MFCD00161522 | 100UG
eMolecules 7-Fluoro-2,3,4,9-tetrahydro-1H-beta-carboline | 177858-80-9 | 250MG | Purity: 95%
Matrix Scientific | 7-Fluoro-2,3,4,9-tetrahydro-1H-beta-carboline | 250MG | 177858-80-9 | MFCD09264527
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eMolecules ChemScene / 1H-Pyrazole-4-carboxamide / 250mg / 654750293 / CS-0205772 / 0.000 / 437701-80-9 / MFCD10001535 / 111.104 / C4H5N3O
ChemScene / 1H-Pyrazole-4-carboxamide / 250mg / 654750293 / CS-0205772 / 0.000 / 437701-80-9 / MFCD10001535 / 111.104 / C4H5N3O
eMolecules Ambeed / 2-(9H-Carbazol-9-yl)acetic acid / 100mg / 552528265 / A109091 / / 524-80-1 / MFCD00439433 / 225.247 / C14H11NO2
Ambeed / 2-(9H-Carbazol-9-yl)acetic acid / 100mg / 552528265 / A109091 / / 524-80-1 / MFCD00439433 / 225.247 / C14H11NO2
Sigma Aldrich Fine Chemicals Biosciences K-252a Ready Made Solution, from Nonomuraea longicatena, >98% | Purity: >98% | Mol Wt: 467.47 | 99533-80-9 | MFCD00161522 | 200UL
K-252a Ready Made Solution, from Nonomuraea longicatena, >98% | Purity: >98% | Mol Wt: 467.47 | 99533-80-9 | MFCD00161522 | 200UL
Medchemexpress LLC Methyl 9H-xanthene-9-carboxylate | 39497-06-8 | 95.0% | C15H12O3 | 250 MG
Methyl 9H-xanthene-9-carboxylate (Methyl xanthanoate) is a drug intermediate used for the synthesis of various active compounds.
- Drug intermediate
- Used for the synthesis of various active compounds
- Appearance: light yellow to yellow oil
- Stable under recommended storage conditions
- Long-term storage for pure form: -20°C for 3 years; 4°C for 2 years
- Storage in solvent: -80°C for 6 months; -20°C for 1 month
Medchemexpress LLC ML339 | 2579689-83-9 | 99.9% | 5 MG
ML339 (CAS 2579689-83-9) is a selective antagonist of the chemokine receptor CXCR6 used in receptor signaling and prostate cancer research. It is supplied as a high-purity solid and has been characterized in functional assays showing nanomolar activity against human CXCR6.
- Selective CXCR6 antagonist (IC50 140 nM).
- Active in human β-arrestin and cAMP assays (0.3 μM and 1.4 μM).
- Markedly less active at mouse CXCR6 (IC50 18 μM).
- High supplied purity (99.88%) and solid powder form.
- Recommended storage: powder -20°C (long term), 4°C (short term); in solvent -80°C.
- Molecular weight 502.00; formula C26H32ClN3O5.
Medchemexpress LLC N2,N6-bis(((9H-fluoren-9-yl)methoxy)carbonyl)-D-lysine | 75932-02-4 | 95.7% | 590.66 g/mol | C36H34N2O6 | 100 G
N2,N6-Bis(((9H-fluoren-9-yl)methoxy)carbonyl)-D-lysine is an Fmoc-protected D-lysine derivative used as a building block in peptide synthesis and other organic synthesis applications.
- Fmoc-protected D-lysine derivative suitable for peptide synthesis.
- Purity 95.7% as supplied.
- Molecular formula C36H34N2O6; molecular weight 590.66 g/mol.
- Appearance: white to off-white solid.
- Storage: powder at -20°C (3 years) or 4°C (2 years); in solvent at -80°C (6 months) or -20°C (1 month).
- Available in gram-scale quantities including 100 G.
Medchemexpress LLC (2S,4R)-1-((9H-Fluoren-9-yl)methyl) 2-methyl 4-hydroxypyrrolidine-1,2-dicarboxylate | 122350-59-8 | C21H21NO5 | 10 G
(2S,4R)-1-((9H-Fluoren-9-yl)methyl) 2-methyl 4-hydroxypyrrolidine-1,2-dicarboxylate is a proline derivative recognized as a beneficial ergogenic dietary substance. It is used as an ergogenic supplement, influencing anabolic hormone secretion, supplying fuel during exercise, enhancing mental performance, and preventing exercise-induced muscle damage.
- Influences anabolic hormone secretion
- Supplies fuel during exercise
- Enhances mental performance during stress-related tasks
- Prevents exercise-induced muscle damage
- Stable as powder at -20°C for 3 years and 4°C for 2 years
- Stable in solvent at -80°C for 6 months and -20°C for 1 month
Medchemexpress LLC (2S,4R)-1-((9H-Fluoren-9-yl)methyl) 2-methyl 4-hydroxypyrrolidine-1,2-dicarboxylate | 122350-59-8 | C21H21NO5 | 100 G
(2S,4R)-1-((9H-Fluoren-9-yl)methyl) 2-methyl 4-hydroxypyrrolidine-1,2-dicarboxylate is a proline derivative with commercial applications as an ergogenic supplement. It influences anabolic hormone secretion, supplies fuel during exercise, impacts mental performance during stressful tasks, and prevents exercise-induced muscle damage.
- Proline derivative
- Influences anabolic hormone secretion
- Supplies fuel during exercise
- Impacts mental performance during stressful tasks
- Prevents exercise-induced muscle damage
- Store as powder at -20°C for up to 3 years or 4°C for up to 2 years
- Store in solvent at -80°C for up to 6 months or -20°C for up to 1 month
- Soluble in DMSO at 100 mg/mL (272.18 mM)