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Filtered Search Results
Medchemexpress LLC Bay 61-3606 hydrochloride | 1615197-10-8 | 98.08% | C20H19ClN6O3 | 5 MG
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BAY 61-3606 hydrochloride is an orally available, ATP-competitive, reversible and highly selective Syk inhibitor with a Ki of 7.5 nM and an IC50 of 10 nM. It reduces ERK1/2 and Akt phosphorylation in neuroblastoma cells and induces a large decrease of Syk phosphorylation in K-rn cell lysates. This compound also sensitizes TRAIL-induced apoptosis by downregulating Mcl-1 in breast cancer cells.
- Orally available
- ATP-competitive and reversible
- Highly selective Syk inhibitor
- Reduces ERK1/2 and Akt phosphorylation in neuroblastoma cells
- Induces a large decrease of Syk phosphorylation in K-rn cell lysates
- Sensitizes TRAIL-induced apoptosis by downregulating Mcl-1 in breast cancer cells
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Medchemexpress LLC RTI-13951-33 hydrochloride | 98.6% | 532.50 | 100 MG
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RTI-13951-33 hydrochloride is a potent, selective, and brain-penetrant GPR88 agonist with an EC50 of 25 nM in a GPR88 cAMP functional assay. This compound reduces alcohol reinforcement and intake behaviors in rats.
- Potent, selective, and brain-penetrant GPR88 agonist.
- Displays an EC50 of 25 nM in GPR88 cAMP functional assay.
- Elevates [35S]-GTPγS binding (EC50, 535 nM) in mouse striatal membranes, but not in membranes from GPR88 knockout mice.
- Exhibits weak affinities at kappa opioid receptor (KOR; Ki, 2.29 μM) and vesicular monoamine transporter (VMAT; Ki, 4.23 μM).
- Shows sufficient brain penetration with a half-life (t1/2) of 48 minutes in rat plasma and 87 minutes in rat brain.
- Dose-dependently decreases alcohol lever responses in a rat model of alcohol self-administration.
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Medchemexpress LLC Seltorexant hydrochloride | 1293284-49-7 | 99.9% | 443.91 | 50 MG
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Seltorexant hydrochloride (JNJ-42847922 hydrochloride) is an orally active, high-affinity, and selective OX2R antagonist (pKi values of 8.0 and 8.1 for human and rat OX2R). It crosses the blood-brain barrier and quickly occupies OX2R binding sites in the rat brain. It is for research use only.
- Orally active
- High-affinity and selective OX2R antagonist
- Crosses the blood-brain barrier
- Quickly occupies OX2R binding sites in the rat brain
- Dose-dependently induces and prolongs sleep in male Sprague-Dawley rats
- Sleep-promoting effects are maintained upon 7-day repeated dosing in rats
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Medchemexpress LLC GSK 1562590 hydrochloride | 1003878-07-6 | 99.0% | 617.95 | 10 MG
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GSK 1562590 hydrochloride is a high-affinity and selective antagonist of the urotensin-II receptor (UT), with pKis ranging from 9.14 to 9.66 for mammalian recombinant (mouse, rat, cat, monkey, human) and native UT. It is intended for research use only.
- High affinity and selective antagonist of urotensin-II receptor (UT).
- PKis of 9.14-9.66 for mammalian recombinant (mouse, rat, cat, monkey, human) and native UT.
- Appears as a solid, white to off-white in color.
- Soluble in DMSO (25 mg/mL).
- Storage recommendations: -20°C, protect from light, stored under nitrogen; in solvent: -80°C for 6 months; -20°C for 1 month.
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Medchemexpress LLC Amisulpride hydrochloride | 81342-13-4 | MFCD00958763 | 99.8% | C17H28ClN3O4S | 100 MG
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Amisulpride hydrochloride is a dopamine D2/D3 receptor antagonist, characterized by Kis of 2.8 and 3.2 nM for human dopamine D2 and D3 receptors, respectively. This compound is widely utilized in pharmacological research to investigate dopamine receptor activity and its associated physiological effects.
- Dopamine D2/D3 receptor antagonist
- Kis of 2.8 and 3.2 nM for human dopamine D2 and D3
- Inhibits quinpirole-elicited [3H]thymidine incorporation
- Increases [3H]dopamine release from rat striatum slices
- Used in studies related to neurological and neurodegenerative diseases
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Medchemexpress LLC Tracazolate hydrochloride | 1135210-68-2 | 99.2% | 5 MG
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Tracazolate (ICI 136753) hydrochloride is a potent GABAA receptor modulator with selectivity for β3, exhibiting anxiolytic and anticonvulsant activity. Its potency is determined by the nature of the third subunit (γ1-3, δ, ε) within the receptor complex. This compound is for research use only and not sold to patients.
- Potentiates α1β1γ2s (EC50=13.2 μM) and α1β3γ2 (EC50=1.5 μM).
- Inhibits α1β1ε (EC50=4.0 μM), α1β3ε (EC50=1.2 μM), α1β3 (EC50=2.7 μM), and α6β3γ (EC50=1.1 μM).
- Interacts with γ-aminobutyric acid GABAA receptors, adenosine receptors, and phosphodiesterases.
- Increases maximum current amplitude and enhances sensitivity of α1β2δ-containing GABAA receptors in oocytes at 10 μM.
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Medchemexpress LLC Desipramine hydrochloride | 58-28-6 | 99.8% | 500 MG
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Desipramine hydrochloride is an inhibitor of norepinephrine transporter (NET), 5-HT transporter (SERT), and dopamine transporter (DAT) with Ki values of 4, 61, and 78,720 nM, respectively. It is intended for research use only.
- Inhibits norepinephrine transporter (NET), 5-HT transporter (SERT), and dopamine transporter (DAT).
- High purity of 99.76%.
- Available in various quantities and formulations (solid, solution in DMSO).
- Used in numerous publications, including studies on cell proliferation/viability, apoptosis-related proteins, and various cellular staining methods.
- Relevant in research areas such as infection, neurological diseases, and cancer.
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Medchemexpress LLC Dapiprazole hydrochloride | 72822-13-0 | 99.3% | C19H28ClN5 | 25 MG
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Dapiprazole hydrochloride is a potent, selective, and orally active alpha-1 adrenoceptor antagonist. It suppresses opioid withdrawal symptoms and is also utilized in eye drops to reverse mydriasis.
- Potent, selective, and orally active alpha-1 adrenoceptor antagonist
- Suppresses opioid withdrawal symptoms
- Used in eye drops for reversing mydriasis
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Medchemexpress LLC 3-MeOARh-NTR | 596.61 | 5 MG
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3-MeOARh-NTR is an activatable imaging probe with high selectivity and good stability, designed for nitroreductase (NTR) detection. It offers a high signal-to-noise ratio, making it an efficient molecular tool for endogenous NTR detection and useful for evaluating kidney hypoxia.
- Produces a strong fluorescence signal in living HeLa cells with decreasing oxygen contents
- Produces fluorescence imaging of kidney tissues from mice with excitation = 488 nm and emission = 510-590 nm
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Medchemexpress LLC Flibanserin | 167933-07-5 | 99.0% | C20H22ClF3N4O.0.5C3H8O.0.5H2O | 100 MG
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Flibanserin hydrochloride (propan-2-ol) hydrate is an orally active compound that acts as a serotonin 5-HT1A receptor agonist and 5-HT2A receptor antagonist, with Ki values of 1 nM and 49 nM respectively. It also interacts with dopamine D4 receptors, showing a Ki value of 4-24 nM.
- Exhibits anti-depression effects.
- Demonstrates anti-anxiety effects.
- Useful for research into hypoactive sexual desire disorder (HSDD).
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Medchemexpress LLC Cefotiam hexetil hydrochloride | 95789-30-3 | 95.1% | C27H39Cl2N9O7S3 | 5 MG
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Cefotiam hexetil hydrochloride (CTM-HE) is an oral third-generation cephalosporin. It acts as a proagent of cefotiam, an antibiotic. While CTM-HE itself lacks anti-bacterial properties, it is intended strictly for research use and is not for sale to patients.
- Oral third-generation cephalosporin
- Proagent of cefotiam
- For research use only
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Medchemexpress LLC Hsp90-IN-17 hydrochloride | 1253584-63-2 | 99.3% | 476.87 | 50 MG
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Hsp90-IN-17 hydrochloride is an HSP90 inhibitor used in the study of proliferative diseases, including cancer and neurodegenerative diseases. It has an IC50 of 0.362 μM against human A2780 cells in an antiproliferative activity assay.
- Can be used in the study of proliferative diseases
- Exhibits antiproliferative activity against human A2780 cells
- Suitable for research use only
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Medchemexpress LLC Resminostat (hydrochloride) | 1187075-34-8 | 99.67% | 385.87 | 25 MG
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Resminostat hydrochloride is a potent inhibitor of HDAC1, HDAC3, and HDAC6, with IC50 values in the nanomolar range. It is used for research applications and appears as a white to off-white solid. This compound shows less potent activity against HDAC8.
- Potent inhibitor of HDAC1, HDAC3, and HDAC6
- Exhibits less potent activity against HDAC8
- Induces histone acetylation in myeloma cells
- Inhibits cell growth and induces apoptosis in myeloma cells
- Synergistic activity with anti-myeloma agents
- Reduces viability of HCC cells when co-treated with AZD-2014
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Medchemexpress LLC CARM1-IN-3 dihydrochloride | 912970-67-3 | C24H34Cl2N4O2 | 50 MG
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CARM1-IN-3 dihydrochloride (compound 17b) is a potent and selective co-activator associated arginine methyltransferase (CARM1) inhibitor.
- Potent and selective CARM1 inhibitor
- IC50 value of 0.07 μM for CARM1
- IC50 value of >25 μM for CARM3
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Medchemexpress LLC Pat1inh-b01 hydrochloride | C22H19BrClF3N6O2 | 5 MG
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PAT1inh-B01 hydrochloride is a selective SLC26A6 inhibitor that blocks fluid absorption in the small intestine. It can be used for research into small intestinal hyposecretory disorders. For research use only, not for sale to patients.
- Inhibits PAT1 (a Cl-/HCO3- exchanger)-mediated anion exchange with an IC50 of 350 nM
- Blocks fluid absorption in the small intestine
- Suitable for research of small intestinal hyposecretory disorders
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