Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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1,606
Tocris Bioscience™ Brefeldin A
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CAS: 20350-15-6 Molecular Formula: C16H24O4
| CAS | 20350-15-6 |
|---|---|
| Molecular Formula | C16H24O4 |
1,607
Tocris Bioscience™ K 22
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Inhibits coronavirus RNA replication; impairs double membrane vesicle (DMV) formation
| Target | DNA, RNA and Protein Synthesis Inhibitors |
|---|---|
| CAS | 2141978-86-9 |
| Purity | 0.98 |
| Chemical Name or Material | N-[(1 Z)-1-[[4-(4-Bromophenyl)-4-hydroxy-1-piperidinyl]carbonyl]-2-phenylethenyl]benzamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C27H25BrN2O3 |
1,608
Tocris Bioscience™ Thalidomide 4'-ether-alkylC8-amine
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Cereblon ligand with alkyl linker and terminal amine for onward chemistry
1,609
Tocris Bioscience™ VCP 171
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Positive allosteric modulator (PAM) of A1 receptors; also allosteric partial agonist in absence of orthosteric agonist
| Target | Adenosine A1 Receptor Modulators |
|---|---|
| CAS | 1018830-99-3 |
| Purity | 0.98 |
| Chemical Name or Material | [2-Amino-4-[3-(trifluoromethyl)phenyl]-3-thienyl]phenylmethanone |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C18H12F3NOS |
1,610
Tocris Bioscience™ SB 399885 hydrochloride
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CAS: 402713-81-9 Molecular Formula: C18H22Cl3N3O4S
| CAS | 402713-81-9 |
|---|---|
| Molecular Formula | C18H22Cl3N3O4S |
1,611
Tocris Bioscience™ BMS 536924
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CAS: 468740-43-4 Molecular Formula: C25H26ClN5O3
| CAS | 468740-43-4 |
|---|---|
| Molecular Formula | C25H26ClN5O3 |
1,612
Tocris Bioscience™ CGP 54626 hydrochloride
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CAS: 149184-21-4 Molecular Formula: C18H29Cl3NO3P
| CAS | 149184-21-4 |
|---|---|
| Molecular Formula | C18H29Cl3NO3P |
1,613
Tocris Bioscience™ CHPG Sodium salt
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Selective mGlu5 agonist. Sodium salt of CHPG (Cat. No. 1049)
| Inhibitors | CHPG Sodium salt |
|---|---|
| Product Type | CHPG Sodium salt |
| Molecular Weight (g/mol) | 223.59 |
| Purity | >99% |
1,614
Tocris Bioscience™ GSK LSD 1 Dihydrochloride
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Potent and selective LSD1 inhibitor
| CAS | 2102933-95-7 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Solubility | Soluble to 100mM in water and to 100mM in DMSO |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | GSK LSD 1 dihydrochloride |
| Recommended Storage | Store at 4°C |
| Synonym | rel-N-[(1S,2R)-2-Phenylcyclopropyl]-4-piperidinamine dihydrochloride |
| Molecular Formula | C14H20N2·2HCl |
| Formula Weight | 289.24 |
1,615
Tocris Bioscience™ Cardamonin
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CAS: 19309-14-9 Molecular Formula: C16H14O4
| CAS | 19309-14-9 |
|---|---|
| Molecular Formula | C16H14O4 |
1,616
Tocris Bioscience™ (+)-Muscarine iodide
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CAS: 24570-49-8 Molecular Formula: C9H20INO2
| CAS | 24570-49-8 |
|---|---|
| Molecular Formula | C9H20INO2 |
1,617
Tocris Bioscience™ CPCCOEt
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CAS: 179067-99-3 Molecular Formula: C13H13NO4
| CAS | 179067-99-3 |
|---|---|
| Molecular Formula | C13H13NO4 |
1,618
Tocris Bioscience™ Diphenhydramine hydrochloride
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CAS: 147-24-0 Molecular Formula: C17H22ClNO
| CAS | 147-24-0 |
|---|---|
| Molecular Formula | C17H22ClNO |
1,619
| Target | Class I Histone Deacetylases Inhibitors |
|---|---|
| Purity | 98% |
| Chemical Name or Material | N-(2-Aminophenyl)-5-[(phenylmethyl)amino]-2-pyrazinecarboxamide dihydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C18H17N5O.2HCl |
1,620
Tocris Bioscience™ JTE 607 Dihydrochloride
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Cytokine release inhibitor; anti-inflammatory
| CAS | 188791-09-5 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Solubility | Soluble to 100mM in water and to 100mM in DMSO |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | JTE 607 dihydrochloride |
| Recommended Storage | Desiccate at Room Temperature |
| Synonym | N-[3,5-Dichloro-2-hydroxy-4-[2-(4-methyl-1-piperazinyl)ethoxy]benzoyl]-L-phenylalanine ethyl ester dihydrochloride |
| Molecular Formula | C25H31Cl2N3O5·2HCl |
| Formula Weight | 597.36 |