Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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1,906
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1,920
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1,906
R&D Systems™ Vandetanib
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent VEGFR-2 inhibitor, also inhibits EGFR and RET oncoproteins activity
| Target | VEGF Receptor Inhibitors |
|---|---|
| CAS | 443913-73-3 |
| Purity | 0.98 |
| Chemical Name or Material | N-(4-Bromo-2-fluorophenyl)-6-methoxy-7-[(1-methyl-4-piperidinyl)methoxy]-4-quinazolinamine |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C22H24BrFN4O2 |
1,907
R&D Systems™ iBET-BD2
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective pan-BD2 inhibitor; orally bioavailable
| Target | Bromodomain Inhibitors |
|---|---|
| CAS | 2474876-09-8 |
| Purity | 0.98 |
| Chemical Name or Material | 4-(Acetylamino)-3-fluoro-N-(trans-4-hydroxycyclohexyl)-5-[(1 S)-1-phenylethoxy]benzamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C23H27FN2O4 |
1,908
R&D Systems™ NS 1619
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 153587-01-0 Molecular Formula: C15H8F6N2O2
| CAS | 153587-01-0 |
|---|---|
| Molecular Formula | C15H8F6N2O2 |
1,909
R&D Systems™ AG 205
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Progesterone receptor membrane component 1 (Pgrmc1) ligand
| CAS | 442656-02-2 |
|---|---|
| Chemical Name or Material | cis-2-[[1-(4-Chlorophenyl)-1H-tetrazol-5-yl]thio]-1-(1,2,3,4,4a,9b-hexahydro-2,8-dimethyl-5H-pyrido[4,3-b]indol-5-yl)-ethanone |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C22H23ClN6OS |
| Formula Weight | Observed MW: 454.98 |
| Assay Percent Range | >98% |
1,910
R&D Systems™ ASB 14780
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective cytosolic phospholipase A2 alpha (cPLA2α) inhibitor; active in vivo; orally bioavailable
1,911
R&D Systems™ GW 843682X
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 660868-91-7 Molecular Formula: C22H18F3N3O4S
| CAS | 660868-91-7 |
|---|---|
| Molecular Formula | C22H18F3N3O4S |
1,912
R&D Systems™ NU 9056
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 1450644-28-6 Molecular Formula: C6H4N2S4
| CAS | 1450644-28-6 |
|---|---|
| Molecular Formula | C6H4N2S4 |
1,913
R&D Systems™ EMD 527040 hydrochloride
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. ανβ6 integrin inhibitor
1,914
R&D Systems™ CATPB
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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1,915
R&D Systems™ KN 92
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 1135280-28-2 Molecular Formula: C24H28ClN2O7PS
| CAS | 1135280-28-2 |
|---|---|
| Molecular Formula | C24H28ClN2O7PS |
1,916
R&D Systems™ Tolvaptan
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective vasopressin V2 receptor antagonist; renoprotective and orally active
| Inhibitors | Tolvaptan |
|---|---|
| Product Type | Tolvaptan |
| Molecular Weight (g/mol) | 448.94 |
| Purity | >98% |
1,917
R&D Systems™ LG 100268
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective RXR agonist; also activates RXR/PPARγ heterodimers
| CAS | 153559-76-3 |
|---|---|
| Chemical Name or Material | 6-[1-(5,6,7,8-Tetrahydro-3,5,5,8,8-pentamethyl-2-naphthalenyl)cyclopropyl]-3-pyridinecarboxylic acid |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C24H29NO2 |
| Formula Weight | Observed MW: 363.49 |
| Assay Percent Range | >98% |
1,918
R&D Systems™ SID 7969543
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 868224-64-0 Molecular Formula: C24H24N2O7
| CAS | 868224-64-0 |
|---|---|
| Molecular Formula | C24H24N2O7 |
1,919
R&D Systems™ (+)-Clopidogrel hydrogen sulfate
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 120202-66-6 Molecular Formula: C16H18ClNO6S2
| CAS | 120202-66-6 |
|---|---|
| Molecular Formula | C16H18ClNO6S2 |
1,920
R&D Systems™ NBOH-2C-CN hydrochloride
A Tocris product, part of R&D Systems. High affinity, selective 5-HT2A agonist
| Inhibitors | NBOH-2C-CN hydrochloride |
|---|---|
| Product Type | NBOH-2C-CN hydrochloride |
| Molecular Weight (g/mol) | 348.82 |
| Purity | >98% |