Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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2,161
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2,175
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60,549
results
2,161
R&D Systems™ Sacubitril calcium
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Membrane metallo-endopeptidase (neprilysin) inhibitor prodrug; orally bioavailable
| Target | Additional Synthetic Protease Inhibitors |
|---|---|
| CAS | 1369773-39-6 |
| Purity | >98% |
| Chemical Name or Material | Ethyl (αR,γS)-γ-[(3-carboxy-1-oxopropyl)amino]-α-methyl-[1,1′-biphenyl]-4-pentanoate hemicalcium salt |
| Recommended Storage | Store at -20°C |
| Synonym | AHU 377 |
| Molecular Formula | C24H28NO5.1/2Ca |
| Formula Weight | 430.52 |
2,162
R&D Systems™ CCMI
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 917837-54-8 Molecular Formula: C19H15Cl2N3O2
| CAS | 917837-54-8 |
|---|---|
| Molecular Formula | C19H15Cl2N3O2 |
2,163
R&D Systems™ Thalidomide 4'-ether-alkylC2-amine
A Tocris product, part of R&D Systems. Cereblon ligand with alkyl linker and terminal amine for onward chemistry
2,164
R&D Systems™ TEPP 46
A Tocris product, part of R&D Systems. Potent and selective pyruvate kinase M2 (PKM2) allosteric activator
| Target | PKM2 |
|---|---|
| CAS | 1221186-53-3 |
| Purity | 0.98 |
| Chemical Name or Material | 6-[(3-Aminophenyl)methyl]-4,6-dihydro-4-methyl-2-(methylsulfinyl)-5H-thieno[2',3':4,5]pyrrolo[2,3-d]pyridazin-5-one |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C17H16N4O2S2 |
2,165
R&D Systems™ UNC 6934
A Tocris product, part of R&D Systems. Antagonizes PWWP1 interaction with nucleosomal H3K36me2, alters NSD2 nucleolar localization
| Target | Lysine Methyltransferase Inhibitors |
|---|---|
| CAS | 2561494-77-5 |
| Chemical Name or Material | N-Cyclopropyl-3,4-dihydro-3-oxo-N-[[4-[(4-pyrimidinylamino)carbonyl]phenyl]methyl]-2H-1,4-benzoxazine-7-carboxamide |
| Molecular Formula | C24H21N5O4 |
2,166
R&D Systems™ Trolox
A Tocris product, part of R&D Systems. Antifade reagent; antioxidant vitamin E derivative; cell permeable and water soluble
2,167
| Target | Sphingosine-1-phosphate Receptor Agonists |
|---|---|
| CAS | 1449747-00-5 |
| Purity | 0.99 |
| Chemical Name or Material | 1-[2-[2,5-Dimethyl-1-(phenylmethyl)-1H-pyrrol-3-yl]-2-oxoethyl]-1,6-dihydro-6-oxo-3-pyridinecarbonitrile |
| Recommended Storage | Store at +4°C |
| Molecular Formula | C21H19N3O2 |
2,168
R&D Systems™ Evofosfamide
A Tocris product, part of R&D Systems. Hypoxia-activated DNA alkylating agent prodrug
| Target | Apoptosis Inducer Compounds |
|---|---|
| CAS | 918633-87-1 |
| Purity | 0.98 |
| Chemical Name or Material | (1-Methyl-2-nitro-1H-imidazol-5-yl)methyl N,N'-bis(2-bromoethyl)phosphorodiamidate |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C9H16Br2N5O4P |
2,169
R&D Systems™ NH 125
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 278603-08-0 Molecular Formula: C27H45IN2
| CAS | 278603-08-0 |
|---|---|
| Molecular Formula | C27H45IN2 |
2,170
R&D Systems™ PIPE 3297 dihydrochloride
A Tocris product, part of R&D Systems. Potent and selective κ opioid receptor agonist; devoid of β-Arrestin-2 recruitment. Also induces differentiation of OPC.
2,171
R&D Systems™ Selinexor
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Selective exportin 1 (XPO1/CRM1) inhibitor
| Target | Antiviral Compounds |
|---|---|
| CAS | 1393477-72-9 |
| Chemical Name or Material | (2Z)-3-[3-[3,5-Bis(trifluoromethyl)phenyl]-1H-1,2,4-triazol-1-yl]-2-propenoic acid 2-(2-pyrazinyl)hydrazide |
| Recommended Storage | Store the unopened product at -20 to -70 °C. Use a manual defrost freezer and avoid repeated freeze-thaw cycles. Do not use past expiration date. |
| Molecular Formula | C17H11F6N7O |
2,172
R&D Systems™ TC-E 5002
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Selective KDM2/7 inhibitor
| Inhibitors | TC-E 5002 |
|---|---|
| Product Type | TC-E 5002 |
| Molecular Weight (g/mol) | 285.38 |
| Purity | >98% |
2,173
R&D Systems™ Clotrimazole
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 23593-75-1 Molecular Formula: C22H17ClN2
| CAS | 23593-75-1 |
|---|---|
| Molecular Formula | C22H17ClN2 |
2,174
R&D Systems™ Pomalidomide 4'-PEG1-acid
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Cereblon ligand with PEG linker and terminal acid for onward chemistry
2,175
R&D Systems™ SGC 6870N
A Tocris product, part of R&D Systems. Negative control for SGC 6870 (Cat. No. 7182)
| Target | Protein Arginine Methyltransferase Inhibitors |
|---|---|
| CAS | 2561471-15-4 |
| Purity | 0.98 |
| Chemical Name or Material | (S)-4-(5-Bromothiophene-2-carbonyl)-5-(3,5-dimethylphenyl)-7-methyl-1,3,4,5-tetrahydro-2H-benzo[e][1,4]diazepin-2-one |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C23H21BrN2O2S |