Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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241
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241
Tocris Bioscience™ DSRM-3716
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and reversible SARM1 NAD hydrolase inhibitor
243
Nutlin-3, Thermo Scientific™
CAS: 548472-68-0 Molecular Formula: C30 H30 Cl2 N4 O4 Molecular Weight (g/mol): 581.49 InChI Key: BDUHCSBCVGXTJM-UHFFFAOYNA-N IUPAC Name: 4-[4,5-bis(4-chlorophenyl)-2-[4-methoxy-2-(propan-2-yloxy)phenyl]-4,5-dihydro-1H-imidazole-1-carbonyl]piperazin-2-one SMILES: COC1=CC=C(C2=NC(C(N2C(=O)N2CCNC(=O)C2)C2=CC=C(Cl)C=C2)C2=CC=C(Cl)C=C2)C(OC(C)C)=C1
| CAS | 548472-68-0 |
|---|---|
| Molecular Weight (g/mol) | 581.49 |
| SMILES | COC1=CC=C(C2=NC(C(N2C(=O)N2CCNC(=O)C2)C2=CC=C(Cl)C=C2)C2=CC=C(Cl)C=C2)C(OC(C)C)=C1 |
| IUPAC Name | 4-[4,5-bis(4-chlorophenyl)-2-[4-methoxy-2-(propan-2-yloxy)phenyl]-4,5-dihydro-1H-imidazole-1-carbonyl]piperazin-2-one |
| InChI Key | BDUHCSBCVGXTJM-UHFFFAOYNA-N |
| Molecular Formula | C30 H30 Cl2 N4 O4 |
244
Tocris Bioscience™ a-Synuclein Degrader 2bn
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Negative control for α Synuclein Degrader 2b (Cat. No. 8040)
245
Tocris Bioscience™ XMU MP 1
Greener Choice
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and selective ATP-competitive mammalian sterile 20-like kinase (MST) 1/2 inhibitor
246
Tocris Bioscience™ GW 280264X
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent ADAM10 and ADAM17 inhibitor
| Target | Synthetic Metalloprotease Inhibitors |
|---|---|
| CAS | 866924-39-2 |
| Purity | 0.98 |
| Chemical Name or Material | Phenylmethyl N-[(5 S)-5-[[(2 R,3 S)-3-(formylhydroxyamino)-2-(2-methylpropyl)-1-oxohexyl]amino]-6-oxo-6-(2-thiazolylamino)hexyl]carbamate |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C28H41N5O6S |
247
| CAS | 80382-23-6 |
|---|---|
| Molecular Formula | C15H17NaO3 |
248
Tocris Bioscience™ BMH 21
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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RNA polymerase I inhibitor; also p53 pathway activator
| Target | RNA/DNA Polymerase Inhibitors |
|---|---|
| CAS | 896705-16-1 |
| Purity | 98% |
| Chemical Name or Material | N-[2-(Dimethylamino)ethyl]-12-oxo-12 H-benzo[g]pyrido[2,1-b]quinazoline-4-carboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C21H20N4O2 |
| Formula Weight | 360.41 |
249
Tocris Bioscience™ NNMTi
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Nicotinamide N-methyltransferase (NNMT) inhibitor; promotes myoblast differentiation
| CAS | 42464-96-0 |
|---|---|
| Purity | 97% |
| Chemical Name or Material | 5-Amino-1-methylquinolinium iodide |
| Molecular Formula | C10H11IN2 |
250
Tocris Bioscience™ ABT 594 Hydrochloride
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Selective α4β2 nAChR agonist
| CAS | 203564-54-9 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | (R)-5-(Azetidin-2-ylmethoxy)-2-chloropyridine hydrochloride |
| Recommended Storage | Store at -20°C |
| Synonym | Tebanicline |
| Molecular Formula | C9H11ClN2O.HCL |
| Formula Weight | 235.11 |
251
Tocris Bioscience™ Neratinib
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent HER2 receptor tyrosine kinase and EGFR kinase inhibitor
| Target | EGF Receptor Inhibitors |
|---|---|
| CAS | 698387-09-6 |
| Purity | 0.98 |
| Chemical Name or Material | (2 E)-N-[4-[[3-Chloro-4-(2-pyridinylmethoxy)phenyl]amino]-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-2-butenamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C30H29ClN6O3 |
252
Tocris Bioscience™ LP 922056
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Notum inhibitor; activates Wnt signaling
| CAS | 1365060-22-5 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 2-[(6-Chloro-7-cyclopropylthieno[3,2-d]pyrimidin-4-yl)thio]acetic acid |
| Molecular Formula | C11H9ClN2O2S2 |
253
Tocris Bioscience™ PLpro inhibitor 6
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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SARS-CoV and SARS-CoV-2 PLpro inhibitor
| Target | Papain-like Protease Inhibitors |
|---|---|
| CAS | 1093070-14-4 |
| Purity | 0.98 |
| Chemical Name or Material | 5-(Acetylamino)-2-methyl-N-[(1 R)-1-(1-naphthalenyl)ethyl]benzamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C22H22N2O2 |
254
Tocris Bioscience™ dTAG-Fluorescein
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Fluorescent probe for labeling mutant FKBP12F36V proteins
255
| CAS | 5234-68-4 |
|---|---|
| Molecular Formula | C12H13NO2S |