Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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556
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570
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60,533
results
556
R&D Systems™ MYX 1715
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. N-myristoyltransferase (NMT) inhibitor
557
R&D Systems™ DCLK1-IN-1
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective doublecortin like kinase 1/2 (DCLK1/2) inhibitor; orally bioavailable
558
R&D Systems™ TM 38837
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Highly potent CB1 inverse agonist; peripherally restricted
559
R&D Systems™ RU.521
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective inhibitor of cyclic GMP-AMP synthase (cGAS)
| Target | Synthase/Synthetase Inhibitors |
|---|---|
| CAS | 2262452-06-0 |
| Purity | 0.98 |
| Chemical Name or Material | 3-[1-(6,7-Dichloro-1 H-benzimidazol-2-yl)-5-hydroxy-3-methyl-1 H-pyrazol-4-yl]-1(3 H)-isobenzofuranone |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C19H12Cl2N4O3 |
560
R&D Systems™ Pomalidomide 4'-alkylC2-azide
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Cereblon ligand with alkyl linker and terminal azide for onward chemistry
561
R&D Systems™ TL 13-22
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Negative control for TL 13-12
562
R&D Systems™ Dooku 1
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Reversibly blocks Yoda1 activity; does not affect constitutive Piezo1 activity
| Target | Other Piezo Channel Compounds |
|---|---|
| CAS | 2253744-54-4 |
| Purity | 98% |
| Chemical Name or Material | 2-[(2,6-Dichlorobenzyl)thio)-5-(1 H-pyrrol-2-yl)-1,3,4-oxadiazole |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C13H9Cl2N3OS |
| Formula Weight | 326.2 |
563
R&D Systems™ KYP 2047
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. High affinity prolyl oligopeptidase inhibitor (Ki = 0.023 nM); anti-angiogenic, neuroprotective and brain penetrant
| CAS | 796874-99-2 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | (2S)-1-[[(2S)-1-(1-Oxo-4-phenylbutyl)-2-pyrrolidinyl]carbonyl]-2-pyrrolidinecarbonitrile |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C20H25N3O2 |
| Formula Weight | 339.44 |
564
R&D Systems™ ML T7
A Tocris product, part of R&D Systems. Inhibitor of phosphatidylserine/CEACAM1 binding to Tim-3
| Target | CEACAM1/CD66a |
|---|---|
| CAS | 459789-75-4 |
| Purity | 0.98 |
| Chemical Name or Material | 5-(2,4-Dichlorophenyl)-3a,6a-dihydro-3-(4-methylphenyl)spiro[1H-furo[3,4-c]pyrrole-1,2'-[2H]indene]-1',3',4,6(3H,5H)-tetrone |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C27H17Cl2NO5 |
565
R&D Systems™ Pomalidomide 4'-PEG4-acid
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Cereblon ligand with PEG linker and terminal acid for onward chemistry
566
R&D Systems™ GSK 9311 Hydrochloride
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Negative control for GSK 6853
| Purity | 98% |
|---|---|
| Chemical Name or Material | N-[2,3-Dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-N-ethyl-2-methoxybenzamide hydrochloride |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C24H31N5O3.HCl |
| Formula Weight | 474 |
567
R&D Systems™ LY 2603618
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective Chk1 inhibitor (IC50 = 7 nM)
| CAS | 911222-45-2 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | N-[5-Bromo-4-methyl-2-[(2S)-2-morpholinylmethoxy)phenyl]-N'-(5-methyl-2-pyrazinyl)urea |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C18H22BrN5O3 |
| Formula Weight | 436.3 |
568
R&D Systems™ JT010
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective TRPA1 channel activator (EC50 = 65 nM)
| CAS | 917562-33-5 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 2-Chloro-N-[4-(4-methoxyphenyl)-2-thiazolyl]-N-(3-methoxypropyl)acetamide |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C16H19ClN2O3S |
| Formula Weight | 354.85 |
569
R&D Systems™ HHP 9
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. BET bromodomain Degrader (PROTAC™); also potent Hedgehog pathway inhibitor
570
R&D Systems™ BTD
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Selective TRPC5 activator
| CAS | 896684-04-1 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 6-Methyl-N-[3-(tricyclo[3.3.1.13,7]dec-1-yloxy)propyl]-4H-1,2,4-benzothiadiazine-3-propanamide-1,1-dioxide |
| Molecular Formula | C24H33N3O4S |