Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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Thermo Scientific Chemicals Olaparib
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Thermo Scientific Chemicals Olaparib
CAS: 763113-22-0 Molecular Formula: C24H23FN4O3
| CAS | 763113-22-0 |
|---|---|
| Molecular Formula | C24H23FN4O3 |
64
Novus Biologicals™ Imidazoquinoline Resiquimod (R-848), TLR7 and TLR8 ligand
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65
Tocris Bioscience™ Biotin-NAD+
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Biotinylated-NAD+; substrate for ADP-ribosylation
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Carfilzomib, Thermo Scientific™
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Carfilzomib, Thermo Scientific™
CAS: 868540-17-4 Molecular Formula: C40 H57 N5 O7 Molecular Weight (g/mol): 719.92 MDL Number: MFCD11040997 InChI Key: BLMPQMFVWMYDKT-UHFFFAOYNA-N IUPAC Name: 4-methyl-N-(1-{[4-methyl-1-(2-methyloxiran-2-yl)-1-oxopentan-2-yl]carbamoyl}-2-phenylethyl)-2-{2-[2-(morpholin-4-yl)acetamido]-4-phenylbutanamido}pentanamide SMILES: CC(C)CC(NC(=O)C(CCC1=CC=CC=C1)NC(=O)CN1CCOCC1)C(=O)NC(CC1=CC=CC=C1)C(=O)NC(CC(C)C)C(=O)C1(C)CO1
| CAS | 868540-17-4 |
|---|---|
| Molecular Weight (g/mol) | 719.92 |
| MDL Number | MFCD11040997 |
| SMILES | CC(C)CC(NC(=O)C(CCC1=CC=CC=C1)NC(=O)CN1CCOCC1)C(=O)NC(CC1=CC=CC=C1)C(=O)NC(CC(C)C)C(=O)C1(C)CO1 |
| IUPAC Name | 4-methyl-N-(1-{[4-methyl-1-(2-methyloxiran-2-yl)-1-oxopentan-2-yl]carbamoyl}-2-phenylethyl)-2-{2-[2-(morpholin-4-yl)acetamido]-4-phenylbutanamido}pentanamide |
| InChI Key | BLMPQMFVWMYDKT-UHFFFAOYNA-N |
| Molecular Formula | C40 H57 N5 O7 |
67
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Tocris Bioscience™ NVS-STG2
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Tocris Bioscience™ NVS-STG2
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STING agonist, molecular glue that causes oligomerization of STING
| Target | STING Agonists |
|---|---|
| CAS | 3030588-01-0 |
| Purity | 0.98 |
| Chemical Name or Material | 4-((4-(2-(tert-Butyl)-5,5-dimethyl-1,3-dioxan-2-yl)benzyl)amino)-3-methoxybenzoic acid |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C25H33NO5 |
68
Tocris Bioscience™ TL 0259
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Selective and highly potent Fgr and Lyn kinase inhibitor; orally bioavailable
| Purity | 98% |
|---|---|
| Chemical Name or Material | 3-[(6,7-Dimethoxy-4-quinazolinyl)oxy]-N-[4-[(4-ethyl-1-piperazinyl)methyl]-3-(trifluoromethyl)phenyl]-4-methylbenzamide dihydrochloride |
| Molecular Formula | C32H34F3N5O4.2HCl |
69
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Thermo Scientific Chemicals Bedaquiline fumarate
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Thermo Scientific Chemicals Bedaquiline fumarate
CAS: 845533-86-0 Molecular Formula: C36H35BrN2O6
| CAS | 845533-86-0 |
|---|---|
| Molecular Formula | C36H35BrN2O6 |
70
Tocris Bioscience™ SLU-PP-332
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Potent pan-ERR agonist
| Target | Estrogen and Related Receptor Agonists |
|---|---|
| CAS | 303760-60-3 |
| Purity | 0.98 |
| Chemical Name or Material | (E)-4-Hydroxy-N'-(naphthalen-2-ylmethylene)benzohydrazide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C18H14N2O2 |
71
Tocris Bioscience™ Ivacaftor
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Potent and selective CFTR potentiator
| Target | CFTR |
|---|---|
| CAS | 873054-44-5 |
| Purity | 98% |
| Chemical Name or Material | N-[2,4-Bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxo-3-quinolinecarboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C24H28N2O3 |
72
Tocris Bioscience™ EM12-SO2F
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Potent covalent inhibitor of Cereblon
73
Tocris Bioscience™ EM 12-FS
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Molecular glue; induces degradation of NQAT1
| Target | Molecular Glues |
|---|---|
| CAS | 2839138-44-0 |
| Purity | 0.95 |
| Chemical Name or Material | 3-[6-[(Fluorosulfonyl)oxy]-1,3-dihydro-1-oxo-2H-isoindol-2-yl]-2,6-piperidinedione |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C13H11FN2O6S |
74
Tocris Bioscience™ MK 2206 dihydrochloride
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Potent and selective allosteric Akt1, Akt2 and Akt3 inhibitor
| Target | Akt (Protein Kinase B) Inhibitors |
|---|---|
| CAS | 1032350-13-2 |
| Purity | 0.98 |
| Chemical Name or Material | 8-[4-(1-Aminocyclobutyl)phenyl]-9-phenyl-1,2,4-triazolo[3,4-f][1,6]naphthyridin-3(2H)-one dihydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C25H21N5O.2HCl |
75
Tocris Bioscience™ DCLK1-IN-1
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Potent and selective doublecortin like kinase 1/2 (DCLK1/2) inhibitor; orally bioavailable