Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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1,246
Tocris Bioscience™ Zoledronic Acid
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent farnesyl diphosphate (FPP) synthase inhibitor
| CAS | 118072-93-8 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Color | Off-white |
| Solubility | Soluble to 50mM in 1.1eq. NaOH and to 3mM in water |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | Ras GTPase Inhibitors |
| Recommended Storage | Store at 4°C |
| Synonym | [1-Hydroxy-2-(1H-imidazol-1-yl)ethylidene]bisphosphonic acid |
| Molecular Formula | C5H10N2O7P2 |
| Formula Weight | 272.09 |
1,247
Tocris Bioscience™ AMG 837 hemicalcium salt
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Potent free fatty acid receptor 1 (FFA1/GPR40) partial agonist
| CAS | 1291087-14-3 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Color | White |
| Solubility | Soluble to 100mM in DMSO |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | AMG 837 hemicalcium salt |
| Recommended Storage | Store at 4°C |
| Synonym | (βS)-β-1-Propyn-1-yl-4-[[4'-(trifluoromethyl)[1,1'-biphenyl]-3-yl]methoxy]benzenepropanoic acid hemicalcium salt |
| Molecular Formula | C26H20F3O3.?Ca |
| Formula Weight | 457.47 |
1,248
Tocris Bioscience™ Ruthenium Red
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CAS: 11103-72-3 Molecular Formula: Cl6H46N14O2Ru3
| CAS | 11103-72-3 |
|---|---|
| Molecular Formula | Cl6H46N14O2Ru3 |
1,249
Tocris Bioscience™ Saxagliptin hydrochloride
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DPPIV/CD26 Inhibitors
| CAS | 709031-78-7 |
|---|---|
| Purity | 98% |
| Recommended Storage | Store at -20°C |
| Synonym | (1S,3S,5S)-2-[(2S)-Amino(3-hydroxytricyclo[3.3.1.13,7]dec-1-yl)acetyl]-2-azabicyclo[3.1.0]hexane-3-carbonitrile hydrochloride |
| Molecular Formula | C18H25N3O2.HCl |
| Formula Weight | 351.87 |
1,250
Tocris Bioscience™ NDT 9513727
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CAS: 439571-48-9 Molecular Formula: C36H35N3O4
| CAS | 439571-48-9 |
|---|---|
| Molecular Formula | C36H35N3O4 |
1,251
Tocris Bioscience™ Tiplaxtinin
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Plasminogen activator inhibitor-1 (PAI-1) inhibitor
| Target | Additional Synthetic Protease Inhibitors |
|---|---|
| CAS | 393105-53-8 |
| Purity | >98% |
| Chemical Name or Material | α-Oxo-1-(phenylmethyl)-5-[4-(trifluoromethoxy)phenyl]-1H-indole-3-acetic acid |
| Recommended Storage | Store at 4°C |
| Synonym | PAI 039, tiplasinin |
| Molecular Formula | C24H16F3NO4 |
| Formula Weight | 439.38 |
1,252
Tocris Bioscience™ m-3M3FBS
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CAS: 200933-14-8 Molecular Formula: C16H16F3NO2S
| CAS | 200933-14-8 |
|---|---|
| Molecular Formula | C16H16F3NO2S |
1,253
Tocris Bioscience™ EDA-DA
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Unnatural dipeptide building block with alkyne group for functionalizing peptidoglycan
1,254
Tocris Bioscience™ RKI 1447 dihydrochloride
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Potent and selective ROCK inhibitor; antitumor
| Inhibitors | RKI 1447 dihydrochloride |
|---|---|
| CAS | 1782109-09-4 |
| Product Type | RKI 1447 dihydrochloride |
| Molecular Weight (g/mol) | 399.29 |
| Purity | >99% |
1,255
Tocris Bioscience™ E-4031 dihydrochloride
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CAS: 113559-13-0 Molecular Formula: C21H29Cl2N3O3S
| CAS | 113559-13-0 |
|---|---|
| Molecular Formula | C21H29Cl2N3O3S |
1,256
Tocris Bioscience™ SR 57227 hydrochloride
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CAS: 77145-61-0 Molecular Formula: C10H15Cl2N3
| CAS | 77145-61-0 |
|---|---|
| Molecular Formula | C10H15Cl2N3 |
1,257
Tocris Bioscience™ Bosentan
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High affinity dual ETA and ETB receptor antagonist;orally bioavailable
| Target | Non-selective Endothelin Receptor |
|---|---|
| CAS | 147536-97-8 |
| Product Type | Antagonist |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C27H29N5O6S |
| Formula Weight | 551.61g/mol |
1,258
Tocris Bioscience™ ACT 462206
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Potent, dual orexin receptor antagonist
| Inhibitors | ACT 462206 |
|---|---|
| Product Type | ACT 462206 |
| Molecular Weight (g/mol) | 388.48 |
| Purity | >99% |
1,259
Tocris Bioscience™ TC NTR1 17
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Selective non-peptide NTS1 agonist
| Product Type | TC NTR1 17 |
|---|---|
| Molecular Weight (g/mol) | 522.98 |
| Purity | >99% |
1,260
Tocris Bioscience™ Kynurenic acid
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CAS: 492-27-3 Molecular Formula: C10H7NO3
| CAS | 492-27-3 |
|---|---|
| Molecular Formula | C10H7NO3 |