Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ Adenosine Receptor Agonist, NECA
A cell-permeable adenosine analog that acts a potent non-selective agonist of adenosine receptors (Ki = 14 nM, 20 nM
MilliporeSigma™ Calbiochem™ α2-Antiplasmin, Human Plasma
A 452-amino acid glycoprotein present in plasma at about 70 μg/ml.
MilliporeSigma™ Calbiochem™ Apoptosis Inhibitor II, NS3694
The Apoptosis Inhibitor II, NS3694, also referenced under CAS 426834-38-0, controls the biological activity of Apoptosis. This small molecule/inhibitor is primarily used for Cancer applications.
MilliporeSigma™ Calbiochem™ Apigenin
Induces the reversion of transformed phenotypes of v-H-ras-transformed NIH 3T3 cells at low concentration (12.5 μM).
MilliporeSigma™ Calbiochem™ NAE Inhibitor, MLN4924
NAE Inhibitor, MLN4924, CAS 951950-33-7, is an AMP mimetic that forms a NAE-catalyzed NEDD8 adduct, which acts as a tight-binding, ATP-competitive NAE inhibitor (IC50 = 4.7nM).
MilliporeSigma™ Calbiochem™ Cyclophosphamide Monohydrate
A widely used anti-neoplastic agent that also displays immunosuppressant properties.
MilliporeSigma™ Calbiochem™ ATR Inhibitor IV
A cell-permeable phenylpyrazine derivative that acts as a potent, ATP-competitive ( Ki 13nM; IC50/[ATP] = 70 nM/50μM and 128 nM/100μM), ATR-selective inhibitor with much reduced or little potency against 4 related PIKKs
MilliporeSigma™ Calbiochem™ Autocamtide-2 Related Inhibitory Peptide II, Cell-permeable
The Autocamtide-2 Related Inhibitory Peptide II, Cell-permeable controls the biological activity of calmodulin-dependent protein kinase II. This small molecule/inhibitor is primarily used for Phosphorylation and Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Pepstatin A, Penetratin
A Pepstatin A that is ≈75% less potent against Cathespins D/E than PepA in cell-free assays.
MilliporeSigma™ Calbiochem™ InSolution™ PD 98059
InSolution™ PD 98059, CAS 167869-21-8, is a 5mg/mL solution in DMSO. A a cell-permeable, selective and reversible inhibitor of MAP Kinase Kinase (MEK).
MilliporeSigma™ Calbiochem™ PI 3-Kα Inhibitor VIII
The PI 3-Kα Inhibitor VIII controls the biological activity of PI 3-Kα. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ PTP CD45 Inhibitor
The PTP CD45 Inhibitor, also referenced under CAS 345630-40-2, controls the biological activity of PTP CD45. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ PDK1/Akt/Flt Dual Pathway Inhibitor
The PDK1/Akt/Flt Dual Pathway Inhibitor, also referenced under CAS 331253-86-2, controls the biological activity of PDK1/Akt/Flt. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ InSolution™ Rac1 Inhibitor II, Z62954982
The InSolution™ Rac1 Inhibitor II, Z62954982, also referenced under CAS 1090893-12-1, controls the biological activity of Rac1. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Protein Arginine N-Methyltransferase Inhibitor, AMI-1
The Protein Arginine N-Methyltransferase Inhibitor, AMI-1 controls the biological activity of Protein Arginine N-Methyltransferase. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.