Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ Isradipine
A voltage gated calcium channel gating inhibitor of the dihydropyridine class.
MilliporeSigma™ Calbiochem™ Zonisamide
An antiepileptic agent that blocks voltage-dependent Na(+) channels and T-type Ca(2+) channels.
MilliporeSigma™ Calbiochem™ Lamellipodial Growth Promoter, C8N6 BPA Polyamine
A cell-permeable, fast acting, branched polyamine. Induces growth of actin-enriched lamellipodia within minutes without the need for serum cofactors .
MilliporeSigma™ Calbiochem™ InSolution™ Pepstatin A, Synthetic
A 25 μM (10 mg/583 μL) sterile-filtered solution of Pepstatin A, Synthetic in DMSO.
MilliporeSigma™ Calbiochem™ InSolution™ Etomoxir
A 50 mM (2 mg/118 μL) solution of Etomoxir in H2O.
MilliporeSigma™ Calbiochem™ MCT1 Inhibitor, SR13800
A cell-permeable inhibitor of monocarboxylate transporter 1 (MCT1). Blocks the proliferation of Raji Burkitt lymphoma cells expressing MCT1 (EC50 = 5 nM).
MilliporeSigma™ Calbiochem™ MMP-2 Substrate, Fluorogenic
A quenched fluorescence substrate for MMP-2 (gelatinase A; kcat/Km = 3.97 x 105 M-1s-1).
MilliporeSigma™ Calbiochem™ MMP-1/MMP-9 Substrate, Fluorogenic
An excellent quenched fluorescence substrate for MMP-1 and MMP-9.
MilliporeSigma™ Calbiochem™ Melatonin
A hormone that has been postulated as the mediator of photo-induced anti-gonadotropic activity in photoperiodic mammals.
MilliporeSigma™ Calbiochem™ MMP-2 Inhibitor I
The MMP-2 Inhibitor I, also referenced under CAS 10335-69-0, controls the biological activity of MMP-2. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
MilliporeSigma™ Calbiochem™ MMP-13 Substrate, Fluorogenic
A quenched fluorescence substrate for MMP-13 (collagenase-3; kcat/Km = 1.09 x 106 M-1 s-1).
MilliporeSigma™ Calbiochem™ Met Kinase Inhibitor VI, SGX523
The Met Kinase Inhibitor VI, SGX523, also referenced under CAS 1022150-57-7, controls the biological activity of Met Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ MARK/Par-1 Activity Inhibitor, 39621
The MARK/Par-1 Activity Inhibitor, 39621 controls the biological activity of MARK/Par-1. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ 8-Methoxymethyl-3-isobutyl-1-methylxanthine
A cell-permeable selective inhibitor of Ca2+-calmodulin-dependent phosphodiesterase (PDE I; IC50 = 4 μM).
MilliporeSigma™ Calbiochem™ InSolution™ Akt Inhibitor X
The InSolution™ Akt Inhibitor X, also referenced under CAS 925681-41-0, controls the biological activity of Akt. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.