Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ Tamoxifen Citrate
Tamoxifen is a potent synthetic anti-estrogenic agent.
MilliporeSigma™ Calbiochem™ Paroxetine Hydrochloride
Paroxetine Hydrochloride is a very potent uptake inhibitor highly selective for 5-HT transporter.
MilliporeSigma™ Calbiochem™ Caspase Modulator I, 1541
A cell-permeable phenylimidazopyridinyl-methoxy coumarin compound that inhibits caspase-3 and caspase-6 activities (IC50 = 35 and 38μM, respectively) by targeting both the large and small subunit active si
MilliporeSigma™ Calbiochem™ MG-132
A cell-permeable, potent, reversible proteasome inhibitor (Ki = 4 nM).
MilliporeSigma™ Calbiochem™ Trequinsin, Hydrochloride
Extremely potent and cell-permeable inhibitor of cGMP-inhibited phosphodiesterase (IC50 = 300 pM) and platelet aggregation in vitro.
MilliporeSigma™ Calbiochem™ MMP-1/MMP-9 Substrate, Fluorogenic
An excellent quenched fluorescence substrate for MMP-1 and MMP-9.
MilliporeSigma™ Calbiochem™ Calpain Inhibitor Set
The Calpain Inhibitor Set controls the biological activity of Calpain. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
MilliporeSigma™ Calbiochem™ InSolution™ Fluvastatin, Sodium Salt
A synthetic, competitive inhibitor of HMG-CoA reductase that acts as anti-hypercholesterolemic agent.
MilliporeSigma™ Calbiochem™ Akt Inhibitor XVIII, SC66
The Akt Inhibitor XVIII, SC66 controls the biological activity of Akt. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ SB 225002
A potent, selective, and competitive antagonist of the G-protein coupled receptor CXCR2 (IL-8RB; IC50 = 22 nM for the inhibition of 125I-IL-8 binding to CXCR2).
MilliporeSigma™ Calbiochem™ TNF-α Antagonist
The TNF-α Antagonist controls the biological activity of TNF-α.
MilliporeSigma™ Calbiochem™ NF-κB Activation Inhibitor
The NF-κB Activation Inhibitor, also referenced under CAS 545380-34-5, controls the biological activity of NF-κB. This small molecule/inhibitor is primarily used for Inflammation/Immunology applications.
MilliporeSigma™ Calbiochem™ AdaAhx3L3VS
A potent, covalent, cell-permeable, irreversible inhibitor of chymotrypsin-like (50-100 nM), trypsin-like (1-5 μM), and PGPH (0.5-1 μM) activities of the 20S proteasome.
MilliporeSigma™ Calbiochem™ p38 MAP Kinase Inhibitor VII, SD-169
The p38 MAP Kinase Inhibitor VII, SD-169, also referenced under CAS 1670-87-7, controls the biological activity of p38 MAP Kinase.