Benzoxazines
TARGETMOL CHEMICALS INC VOROZOLE 5MG
Also available in 1 mg 10 mg 25 mg 50 mg and bulk. Please contact Fisher for quotes. Vorozole (R83842) is an orally active potent and selective nonsteroidal aromatase inhibitor.Vorozole exhibits antitumor activity in vivo and may be used in the study of breast cancer. purity: 99%
TARGETMOL CHEMICALS INC MOVELTIPRIL 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Moveltipril (Moveltipril calcium) is a potent angiotensin-converting enzyme (ACE) inhibitor.Moveltipril is converted to captopril in the body for action. purity: 99%
TARGETMOL CHEMICALS INC JC124 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. JC124 is an inhibitor of NLRP3 Inflammasome and exhibits neuroprotective and anti-inflammatory activities. purity: 98%
TARGETMOL CHEMICALS INC GGTI 2147 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg and bulk. Please contact Fisher for quotes. GGTI 2147 decreased Rac1 activity down-regulated p65 expression and ameliorated OGD/R-induced neuronal apoptosis. purity: 99%
TARGETMOL CHEMICALS INC SB 218795 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. SB 218795 is an effective and selective antagonist of NK3 with a Ki 13 nM for hNK3 which is about 90-fold and 7000-fold selectivity over hNK2 and hNK1. purity: 98%
TARGETMOL CHEMICALS INC SR11237 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. SR11237 is a Pan retinoid X receptor (RXR) agonist. SR11237 causes RXR/RXR homodimers to form and transactivate a reporter gene containing a RXR-response element. purity: 98%
TARGETMOL CHEMICALS INC ER 50891 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 500 mg and bulk. Please contact Fisher for quotes. ER-50891 is a potent retinoic acid receptor alpha (RAR(alpha)) antagonist. er-50891 reduces the inhibitory effect of allosteric retinoic acid and restores osteoblast differentiation induced by bone morphogenetic protein 2. purity: 99%
TARGETMOL CHEMICALS INC SQ22536 25MG
Also available in 5 mg 10 mg 50 mg 100 mg 200 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. SQ22536 (9-(tetrahydrofuran-2-yl)-9h-purin-6-amine) the adenosine analogue 9-(Tetrahydro-2-furyl)adenine inhibited adenylate cyclase activity of crude membrane preparations from catfish (Ictalurus melas) and rat isolated hepatocytes in a non-competitive manner. purity: 98%
TARGETMOL CHEMICALS INC FIPAMEZOLE 5MG
Also available in 50 mg 100 mg and bulk. Please contact Fisher for quotes. Fipamezole is a potent alpha2 adrenergic receptor antagonist that may be useful for studying autonomic dysfunction in Parkinson's disease. purity: 99%
TARGETMOL CHEMICALS INC AMPEROZIDE 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Amperozide (FG 5606) is a diphenylbutylpiperazine atypical antipsychotic which antagonizes 5-HT2A receptors. It inhibits dopamine release and alters the firing of dopaminergic neurons. Investigations regarding the use of the agent revolved primarily around its capability for treating schizophrenia in humans. purity: 99%
TARGETMOL CHEMICALS INC ATC 0175 HYDROCHLORIDE 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 500 mg and bulk. Please contact Fisher for quotes. ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective. ATC 0175 hydrochloride has affinity for MCH1R MCH2R MCH1 5-HT2B receptors and 5-HT1A receptors with IC50s of 13.5 nM >10000 nM 13 nM 9.66 nM and 16.9 nM respectively. ATC 0175 hydrochloride exhibits antidepressant and anxiolytic effects in animal models. aTC 0175 can be used to study depression and/or anxiety disorders. purity: 99%
TARGETMOL CHEMICALS INC ARC 239 DIHYDROCHLORIDE 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. ARC 239 dihydrochloride is a selective (alpha)2B adrenoceptor antagonist (pKD values are 8.8 6.7 and 6.4 at (alpha)2B (alpha)2A and (alpha)2D receptors respectively). purity: 98%
TARGETMOL CHEMICALS INC HNMPA 10MG
Also available in 1 mg 2 mg 5 mg 25 mg 50 mg 100 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. HNMPA is a membrane impermeable inhibitor of insulin receptor tyrosine kinase. HNMPA inhibits tyrosine and serine autophosphorylation by the human insulin receptor. HNMPA exhibits no effect on cyclic AMP-dependent protein kinase or protein kinase C activities. purity: 99%
TARGETMOL CHEMICALS INC AD57 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. AD57 is a potent inhibitor of both c-Src and Abl with IC50 of 0.025 uM and 0.041 uM respectively. purity: 98%
TARGETMOL CHEMICALS INC ESI-09 25MG
Also available in 2 mg 5 mg 10 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. ESI-09 is a new-typel noncyclic nucleotide EPAC antagonist.The IC50 values of ESI-09 for EPAC1 and EPAC2 is 3.2 and 1.4 uM respectively. purity: 99%