Cycloheptathiophenes
Medchemexpress LLC Diroximel fumarate | 1577222-14-0 | MFCD10057039 | >98.0% | 255.22 | C11H13NO6 | 25 MG
Diroximel fumarate is an orally active prodrug of monomethyl fumarate used in research to investigate Nrf2 pathway activation and multiple sclerosis-related pharmacology. The compound is provided with analytical data for identification and formulation of stock solutions.
- Orally active prodrug of monomethyl fumarate.
- Useful for in vitro and in vivo studies of Nrf2-mediated pathways.
- Provided with analytical specifications including CAS, formula, and molecular weight for traceability.
- Available in mg-scale quantities suitable for preclinical research.
Apexbio Technology LLC Rupatadine Fumarate 182349-12-8 10mM (in 1mL Ethanol)
Rupatadine Fumarate (CAS 182349-12-8) is a small molecule antagonist targeting platelet-activating factor receptor (PAFR) and histamine H1 receptor It exhibits binding affinities (K i) of 550 nM at PAFR and 102 nM at the histamine H1 receptor effectively inhibiting signaling mediated by these pathways Through dual antagonism rupatadine fumarate disrupts inflammatory and allergic responses regulated by platelet-activating factor and histamine signaling Currently in Phase 2 clinical development it serves as a valuable pharmacological tool for studying inflammation and allergic conditions
Medchemexpress LLC Ocifisertib fumarate | 1616420-30-4 | 99.3% | 650.72 Da | C37H38N4O7 | 5MG
Ocifisertib fumarate is the fumarate salt of Ocifisertib (CFI-400945), a potent, selective, orally bioavailable inhibitor of polo-like kinase 4 (PLK4) used as a research tool in oncology and cell biology to study centriole duplication and mitotic defects. Reported potency values support activity in biochemical and cellular assays.
Medchemexpress LLC Cevipabulin fumarate | 849550-67-0 | MFCD31813783 | 99.9% | 580.89 g/mol | C22H22ClF5N6O5 | 10 MG
Cevipabulin fumarate is the fumarate salt of a microtubule-active small-molecule antitumor agent supplied for laboratory research use. It inhibits tubulin binding, disrupts microtubule dynamics, and produces cytotoxic effects in human tumor cell lines; supplied as a solid with specified storage conditions for stability.
- Microtubule-active mechanism that disrupts tubulin dynamics.
- High chemical purity suitable for research applications.
- Solid, white to off-white physical form for easy handling and storage.
- Storage conditions provided for solid and solution forms to preserve stability.
- Available in small research pack sizes for preclinical studies.
Medchemexpress LLC Ro 48-8071 Fumarate | 189197-69-1 | 99.1% | 564.44 | 50 MG
Ro 48-8071 Fumarate | 189197-69-1 | 99.1% | 564.44 | 50 MG
Medchemexpress LLC Diethyl fumarate | 623-91-6 | 98.97% | 172.18 | 100 G
Diethyl fumarate is a decomposition product of Malathion 9 (a pesticide) and a reactant in the Diels-Alder reaction. It is a reputed skin irritant and can cause non-immunologic contact urticaria on the skin. When hybridized with Curcumin, Diethyl fumarate can exert neuroprotective effects.
- Reactant in the Diels-Alder reaction.
- Exerts neuroprotective effects in combination with curcumin.
- Available in various quantities (mg, g) and solutions.
- High purity (98.97%).