accessibility menu, dialog, popup

UserName
Viewing profile as user:

Imidazoles

Aromatic organic heterocyclic compounds that consist of a diazole with non-adjacent nitrogen atoms with the formula: C3N2H4.

Filtered Search Results

Products from some of our suppliers do not display in filtered search results. Please clear all filters to see these products.

Narrow Results

Narrow Results

category

brands

  • (6)

special interests

  • (6)
Search Within Results
Keyword Search:
1 – 6 of 6 results
1

Medchemexpress LLC Propargyl-PEG4-Boc | 1355197-66-8 | 316.39 | 100 MG
SDP

Propargyl-PEG4-Boc is a PEG-based PROTAC linker utilized in the synthesis of PROTACs. It functions as a click chemistry reagent, containing an Alkyne group, which allows it to undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules that contain Azide groups.

  • Peg-based PROTAC linker
  • Used in the synthesis of PROTACs
  • Click chemistry reagent
  • Contains an alkyne group
  • Can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with azide-containing molecules

ENCOMPASS_PREFERRED
2

Medchemexpress LLC 2-[4-[[4-hydroxy-3-[2-(4-nitrophenyl)ethynyl]-5-propan-2-ylphenyl]methyl]-3,5-dimethylphenoxy]aceti | 447415-26-1 | 99.4% | C28H27NO6 | 10MG
SDP

NH-3 is an orally active, reversible thyroid hormone receptor (THR) antagonist that inhibits hormone binding and cofactor recruitment; it shows potent THR inhibition (IC50 55 nM) and contains an alkyne group enabling copper-catalyzed azide-alkyne cycloaddition for click chemistry applications.

  • Orally active, reversible thyroid hormone receptor antagonist.
  • Potent THR inhibition with reported IC50 of 55 nM.
  • Contains an alkyne group for copper-catalyzed click chemistry.
  • High purity suitable for research use (≈99.4%).
  • Available as powder and DMSO solution formats for flexibility in assays.
  • Recommended storage conditions provided to preserve stability.

ENCOMPASS_PREFERRED
3

Medchemexpress LLC NH-3 | 447415-26-1 | 99.4% | C28H27NO6 | 50 MG
SDP

NH-3 is an orally active, reversible thyroid hormone receptor (THR) antagonist with an IC50 of 55 nM. It is a derivative of the selective thyromimetic GC-1 and works by inhibiting the binding of thyroid hormones to their receptor, thereby inhibiting cofactor recruitment. Additionally, NH-3 is a click chemistry reagent containing an alkyne group, enabling it to undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules that possess azide groups.

  • Orally active, reversible thyroid hormone receptor antagonist
  • IC50 of 55 nM (THR)
  • Inhibits binding of thyroid hormones to their receptor
  • Click chemistry reagent with alkyne group
  • Enables copper-catalyzed azide-alkyne cycloaddition
  • Modestly decreases heart rate in vivo

ENCOMPASS_PREFERRED
4

Medchemexpress LLC NH-3 | 447415-26-1 | 99.4% | C28H27NO6 | 100 MG
SDP

NH-3 is an orally active, reversible thyroid hormone receptor (THR) antagonist with an IC50 of 55 nM. It is derived from the selective thyromimetic GC-1 and inhibits the binding of thyroid hormones to their receptor and also inhibits cofactor recruitment. NH-3 also functions as a click chemistry reagent, featuring an Alkyne group that can participate in copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

  • Orally active, reversible thyroid hormone receptor antagonist
  • Inhibits thyroid hormone binding to its receptor and cofactor recruitment
  • Functions as a click chemistry reagent
  • Contains an alkyne group for copper-catalyzed azide-alkyne cycloaddition
  • Modestly decreases heart rate in vivo
  • Inhibits tachycardic and TSH suppressant effects in vivo

ENCOMPASS_PREFERRED
5

Medchemexpress LLC (S)-4-(8-Amino-3-(1-(but-2-ynoyl)pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl-d4)benzamide | 2699608-18-7 | >=98.0% | 469.53 | 1 MG
SDP

Acalabrutinib-d4 (ACP-196-d4) is a deuterium labeled Acalabrutinib, an orally active, irreversible, and highly selective second-generation BTK inhibitor. It functions as a click chemistry reagent, containing an Alkyne group that can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

  • Used as a tracer for quantitation during drug development.
  • Serves as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS.
  • Incorporates stable heavy isotopes to affect pharmacokinetic and metabolic profiles.
  • Suitable for research use only.

ENCOMPASS_PREFERRED
6

Medchemexpress LLC Ca inhibitor 1 (GS-6207 analog) | 2189684-45-3 | 99.8% | 958.34 g·mol^-1 | C41H36ClF8N7O5S2 | 10MM 1ML
SDP

CA inhibitor 1 is a synthetic HIV capsid inhibitor and alkyne-containing small molecule supplied as a ready-to-use 10 mM solution in DMSO for research and chemical biology applications, including copper-catalyzed azide-alkyne cycloaddition workflows.

  • Supplied as 10 mM solution in DMSO
  • High purity: 99.8%
  • Molecular weight 958.34 g·mol⁻¹
  • Molecular formula C41H36ClF8N7O5S2
  • Contains terminal alkyne for click chemistry applications
  • Recommended storage: powder -20 °C; in solvent -80 °C for long-term storage

ENCOMPASS_PREFERRED