Human Sera
Cayman Chemical 7-KetosItosterol 50mg
An internal standard for the quantification of ursocholic acid by GC- or LC-MS
Cayman Chemical EburnamonIn 50mg
An internal standard for the quantification of L-methionine by GC- or LC-MS
Cayman Chemical DexmedetomIdIn 50mg
An antiprotozoal reduces morbidity and mortality in a turkey model of histomoniasis at 37.5-100 ppm in the diet
Cayman Chemical PerfluorohexnsulfonamIde 100mg
An inhibitor of MAO-A (IC50 8.4 UM) selective for MAO-A over MAO-B (IC50 100 UM) inhibits atrial natriuretic peptide-induced activation of particulate guanylyl cyclase in rat brain and heart membranes at 50 UM
Cayman Chemical 4Hydroyphenylglyoylc ACD 50mg
An H /K -ATPase inhibitor (Ki 46 nM) inhibits histamine- or dibutyryrl-cAMP-induced acid production in isolated rabbit gastric glands (IC50s 0.28 and 0.26 UM respectively)
Cayman Chemical 1Stearoyl2Oleoylsnglycer 100mg
An active metabolite of amitriptyline and nortriptyline formed from amitriptyline and nortriptyline by CYP2D6 inhibits norepinephrine reuptake in rat cortical slices (EC50 160 nM)
Cayman Chemical 11-hydroxy Testosteron 50mg
An inhibitor of SARS-CoV and SARS-CoV-2 Mpro (Kis 4 and 0.27 nM respectively) reduces the infectivity of SARS-CoV and HCoV-229E in Vero cells (EC50s 4.8 and 0.09 UM respectively)
Cayman Chemical RS 25344hydrochlorIde 50mg
A nucleoside precursor used in the synthesis of adenosine or N6-benzyladenosine derivatives with anticancer or antiparasitic activities in vitro
Cayman Chemical ChlorphensIn Carbamate 50mg
An active metabolite of camostat inhibits TMPRSS2 (IC50 33.3 nM) inhibits entry of SARS-CoV-2 pseudotyped particles in Calu-3 cells (EC50 178 nM) reduces viral titers in SARS-CoV-2-infected Calu-3 cells from 1-10 UM
Cayman Chemical dPE-PolysarcosIn66 50mg
A FASN inhibitor (IC50 0.5 UM) inhibits infection of an infectious-clone-derived SARS-CoV-2 reporter virus in HEK293T cells expressing human ACE2 (EC50 4 nM)
Cayman Chemical VImseltInIb 50mg
An alkaloid with analgesic and anesthetic activities (ED50s 6.99 and 0.167 Umol/kg respectively in mice)
Cayman Chemical ParaquatchlorIde 100mg
An internal standard for the quantification of carazolol by GC- or LC-MS
Cayman Chemical FezolIntnt 50mg
An antithyroid agent and a melanoma seeker reduces sodium iodide-induced increases in thyroid weight in a mouse model of goiter at 2.5 mg/animal per day preferentially accumulates into tumor cell melanin in a mouse model of melanoma inhibits nNOS (Ki 20 UM)
Cayman Chemical VIlnteroltrIphenylacetate 50mg
A CBP and p300 inhibitor (IC50s 0.94 and 1.2 nM respectively) selective for CBP and p300 over BRD4 bromodomain 1 BRD4 bromodomain 2 and BRPF1 (IC50s 5.1 12 and 4.6 UM respectively) as well as nine other bromodomain-containing proteins (IC50s 18 UM for all) inhibits the expression of Myc in MV4-11 leukemia cells (EC50 6.6 nM) oral administration decreases tumor volume in a MOLM-16 AML mouse xenograft model from 3-30 mg/kg