Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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2,176
–
2,190
of
60,549
results
2,176
R&D Systems™ PD 4'-oxyacetic acid
A Tocris product, part of R&D Systems. Functionalized cereblon ligand for PROTAC development
2,177
R&D Systems™ Mpro 13b-H
A Tocris product, part of R&D Systems. Negative control for Mpro 13b-K (Cat. No. 7228)
2,178
R&D Systems™ DG 041
A Tocris product, part of R&D Systems. Potent and selective EP3 antagonist; antiplatelet and antithrombotic
| Target | Prostanoid Receptor Antagonists |
|---|---|
| CAS | 861238-35-9 |
| Purity | 0.98 |
| Chemical Name or Material | (2E)-3-[1-[(2,4-Dichlorophenyl)methyl]-5-fluoro-3-methyl-1H-indol-7-yl]-N-[(4,5-dichloro-2-thienyl)sulfonyl]-2-propenamide |
| Recommended Storage | Store at +4°C |
| Molecular Formula | C23H15Cl4FN2O3S2 |
2,179
R&D Systems™ c-Di-AMP sodium salt
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Endogenous STING and DDX41 agonist; activates STING-dependent signaling
2,180
R&D Systems™ 1A-116
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Rac1 inhibitor; blocks Rac1-P-Rex1 interaction
| CAS | 1430208-73-3 |
|---|---|
| Product Type | Inhibitor |
| Purity | 98% |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C16H16F3N3 |
| Formula Weight | 307.31 |
2,181
R&D Systems™ CHDI 00484077
A Tocris product, part of R&D Systems. Potent and selective HDAC class IIa inhibitor
2,182
R&D Systems™ Biotin-PEG4-Diazirine
A Tocris product, part of R&D Systems. Photo-crosslinking capture probe for deazaflavin-diazirine energy-transfer labelling (DarT labelling) with a biotin handle
2,183
R&D Systems™ MKT 077
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 147366-41-4 Molecular Formula: C21H22ClN3OS2
| CAS | 147366-41-4 |
|---|---|
| Molecular Formula | C21H22ClN3OS2 |
2,184
R&D Systems™ AZ PFKFB3 67, >98%
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 1704741-11-6 Molecular Formula: C26H25N5O3
| CAS | 1704741-11-6 |
|---|---|
| Molecular Formula | C26H25N5O3 |
2,185
R&D Systems™ CIM 0216
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Selective TRPM3 agonist
| Target | TRPM Agonists |
|---|---|
| CAS | 1031496-06-6 |
| Purity | >98% |
| Chemical Name or Material | 3,4-Dihydro-N-(5-methyl-3-isoxazolyl)-α-phenyl-1(2H)-quinolineacetamide |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C21H21N3O2 |
| Formula Weight | 347.41 |
2,186
R&D Systems™ Adaptaquin
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. HIF-prolyl hydroxylase-2 (PHD2) inhibitor; antioxidant
| Target | Hydrolase Inhibitors |
|---|---|
| CAS | 385786-48-1 |
| Purity | >97% |
| Chemical Name or Material | 7-[(4-Chlorophenyl)[(3-hydroxy-2-pyridinyl)amino]methyl]-8-quinolinol |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C21H16ClN3O2 |
| Formula Weight | 377.82 |
2,187
R&D Systems™ XY-06-007
A Tocris product, part of R&D Systems. Potent and selective Degrader of Brd4BD1 L94V fusion proteins
2,188
R&D Systems™ SGC 6870
A Tocris product, part of R&D Systems. Potent and selective PRMT6 allosteric inhibitor
| Target | Protein Arginine Methyltransferase Inhibitors |
|---|---|
| CAS | 2561471-27-8 |
| Purity | 0.98 |
| Chemical Name or Material | (R)-4-(5-Bromothiophene-2-carbonyl)-5-(3,5-dimethylphenyl)-7-methyl-1,3,4,5-tetrahydro-2H-benzo[e][1,4]diazepin-2-one |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C23H21BrN2O2S |
2,189
R&D Systems™ ICG 001
A Tocris product, part of R&D Systems. Inhibits TCF/β-catenin-mediated transcription
| Target | beta-Catenin Inhibitors |
|---|---|
| CAS | 780757-88-2 |
| Purity | 0.98 |
| Chemical Name or Material | (6S,9aS)-Hexahydro-6-[(4-hydroxyphenyl)methyl]-8-(1-naphthalenylmethyl)-4,7-dioxo-N-(phenylmethyl)-2H-pyrazino[1,2-a]pyrimidine-1(6H)-carboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C33H32N4O4 |
2,190
R&D Systems™ NS 3861
A Tocris product, part of R&D Systems. α3β2 full agonist; also α3β4 partial agonist
| Target | Additional Nicotinic Receptor Agonists |
|---|---|
| CAS | 216853-60-0 |
| Purity | 0.98 |
| Chemical Name or Material | 3-(3-Bromo-2-thienyl)-8-methyl-8-azabicyclo[3.2.1]oct-2-ene fumarate |
| Recommended Storage | Desiccate at Room Temperature |
| Molecular Formula | C12H14BrNS.C4H4O4 |