Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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1,096
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1,096
Tocris Bioscience™ VU 0357017 hydrochloride
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CAS: 1135242-13-5 Molecular Formula: C18H28ClN3O3
| CAS | 1135242-13-5 |
|---|---|
| Molecular Formula | C18H28ClN3O3 |
1,097
Tocris Bioscience™ CHR 2797
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Aminopeptidase inhibitor
| Inhibitors | CHR 2797 |
|---|---|
| Product Type | CHR 2797 |
| Molecular Weight (g/mol) | 406.48 |
| Purity | >98% |
1,098
Tocris Bioscience™ GS 143
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β-TrCP1 ligase inhibitor
| Target | Ubiquitin Ligase (E3) Inhibitors |
|---|---|
| CAS | 916232-21-8 |
| Purity | >98% |
| Chemical Name or Material | 4-[4-[[5-(2-Fluorophenyl)-2-furanyl]methylene]-4,5-dihydro-5-oxo-3-(phenylmethyl)-1H-pyrazol-1-yl]benzoic acid |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C28H19FN2O4 |
| Formula Weight | 466.46 |
1,099
Tocris Bioscience™ Canertinib dihydrochloride
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Potent EGFR kinase inhibitor
| CAS | 289499-45-2 |
|---|---|
| Chemical Name or Material | N-[4-[(3-Chloro-4-fluorophenyl)amino]-7-[3-(4-morpholinyl)propoxy]-6-quinazolinyl]-2-propenamide dihydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C24H25ClFN5O3.2HCl |
| Formula Weight | Observed MW: 558.86 |
| Assay Percent Range | >98% |
1,100
Tocris Bioscience™ Tomoxetine hydrochloride
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CAS: 82248-59-7 Molecular Formula: C17H22ClNO
| CAS | 82248-59-7 |
|---|---|
| Molecular Formula | C17H22ClNO |
1,101
Tocris Bioscience™ C 176
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mSTING antagonist
| Target | STING Antagonists |
|---|---|
| CAS | 314054-00-7 |
| Purity | 97% |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C11H7IN2O4 |
1,102
Tocris Bioscience™ TAK 165
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Potent and selective ErbB2 inhibitor
| Inhibitors | TAK 165 |
|---|---|
| Product Type | TAK 165 |
| Molecular Weight (g/mol) | 468.47 |
| Purity | >99% |
1,103
Tocris Bioscience™ RA 839
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Nrf2 activator; inhibits Nrf2/Keap1 interaction
| Target | Nrf2 Modulators |
|---|---|
| CAS | 1832713-02-6 |
| Purity | >98% |
| Chemical Name or Material | (3S)-1-[4-[[(2,3,5,6-Tetramethylphenyl)sulfonyl]amino]-1-naphthalenyl]-3-pyrrolidinecarboxylic acid |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C25H28N2O4S |
| Formula Weight | 452.57 |
1,104
Tocris Bioscience™ Liproxstatin-1 hydrochloride
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Additional Apoptosis-related Compounds
| Target | Ferroptosis Inhibitors |
|---|---|
| Purity | 98% |
| Recommended Storage | Store at -20°C |
| Synonym | N-[(3-Chlorophenyl)methyl]spiro[piperidine-4,2′(1′H)-quinoxalin]-3′-amine hydrochloride |
| Molecular Formula | C19H21ClN4.HCl |
| Formula Weight | 377.31 |
1,105
Tocris Bioscience™ XCC
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CAS: 96865-83-7 Molecular Formula: C19H22N4O5
| CAS | 96865-83-7 |
|---|---|
| Molecular Formula | C19H22N4O5 |
1,106
Tocris Bioscience™ PF 06260933 dihydrochloride
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MAP4K4 (HGK) inhibitor; also inhibits MINK and TNIK
| Target | HGK/MAP4K4 |
|---|---|
| CAS | 1883548-86-4 |
| Purity | 98% |
| Chemical Name or Material | 5-(4-Chlorophenyl)-[3,3 '-bipyridine]-6,6 '-diamine dihydrochloride |
| Recommended Storage | Desiccate at Room Temperature |
| Synonym | EC 2.7.11, EC 2.7.11.1, FLH21957, FLJ10410, hepatocyte progenitor kinase-like/germinal center kinase-like kinase, HGKFLJ20373, HPK/GCK-like kinase HGK, KIAA0687, MAP4K4, MAPK/ERK kinase kinase kinase 4, MEK kinase kinase 4, MEKKK 4, MEKKK4, mitogen-activa |
| Molecular Formula | C16H13ClN40.2 HCl |
| Formula Weight | 369.68 |
1,107
Tocris Bioscience™ JH-II-127
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Potent and selective LRRK2 inhibitor
| CAS | 1700693-08-8 |
|---|---|
| Chemical Name or Material | [4-[[5-Chloro-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-3-methoxyphenyl]-4-morpholinyl-methanone |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C19H21ClN6O3 |
| Formula Weight | Observed MW: 416.87 |
| Assay Percent Range | >98% |
1,108
Tocris Bioscience™ XMD 8-92
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CAS: 1234480-50-2 Molecular Formula: C26H30N6O3
| CAS | 1234480-50-2 |
|---|---|
| Molecular Formula | C26H30N6O3 |
1,109
Tocris Bioscience™ TC-S 7009
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High affinity and selective HIF-2α inhibitor
| CAS | 1422955-31-4 |
|---|---|
| Chemical Name or Material | N-(3-Chloro-5-fluorophenyl)-4-nitro-2,1,3-benzoxadiazol-5-amine |
| Recommended Storage | Store at Room Temperature |
| Molecular Formula | C12H6ClFN4O3 |
| Formula Weight | Observed MW: 308.65 |
| Assay Percent Range | >99% |
1,110
Tocris Bioscience™ Tadalafil
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CAS: 171596-29-5 Molecular Formula: C22H19N3O4
| CAS | 171596-29-5 |
|---|---|
| Molecular Formula | C22H19N3O4 |