Cayman Chemical KAT8 InhIbItr 19 10mg
A KAT8 inhibitor; selective for KAT8 over KAT2A, KAT2B, KAT3B, KAT6A, and KAT7 at 200 µM; reduces H4K16Ac in HT-29 cells at 50 µM; reduces the viability of HCT116, H1299, A549, and U937 cancer cells (IC50s = 39.4, 52.1, 41, and 30.1 µM, respectively)