Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ (+/-)-Clopidogrel Hydrogensulfate
A thienopyridine compound that acts as a specific irreversible inhibitor of purinergic P2Y12 recept
MilliporeSigma™ Calbiochem™ Ouabain, Octahydrate
Inhibits Na+,K+-ATPase.
MilliporeSigma™ Calbiochem™ 2-Guanidinoethylmercaptosuccinic Acid
Potent inhibitor of a carboxypeptidase B-like processing enzyme referred to as enkephalin convertase (Ki = 8.8 nM).
MilliporeSigma™ Calbiochem™ Rac1 Inhibitor
Rac1 Inhibitor, CAS 1177865-17-6, is a cell-permeable, reversible inhibitor of Rac1 GDP/GTP exchange. Interferes with the interaction between Rac1 and Rac-specific GEFs Trio and Tiam1 (IC50 ≈50 μM).
MilliporeSigma™ Calbiochem™ Elastase Substrate V, Fluorogenic
Elastase Substrate V, Fluorogenic, CAS 72252-90-5, is a sensitive fluorogenic substrate for the quantitative determination of human leukocyte and porcine pancreatic elastase (Km = 140 μM).
MilliporeSigma™ Calbiochem™ Protease Inhibitor Cocktail Set III, Animal-Free
Protease Inhibitor Cocktail Set III, Animal-Free, is a cocktail of six protease inhibitors with broad specificity for the inhibition of aspartic, cysteine & serine proteases & aminopeptidases.
MilliporeSigma™ Calbiochem™ 12/15-Lipoxygenase Inhibitor, ML351
A cell-permeable, highly potent, selective, active site directed, mixed type inhibitor of lipoxygenase-12/15 (IC50 = 200 nM for human).
MilliporeSigma™ Calbiochem™ 2,3-Butanedione 2-Monoxime
An inhibitor of skeletal and cardiac muscle contraction.
MilliporeSigma™ Calbiochem™ IP6K Inhibitor
The IP6K Inhibitor, also referenced under CAS 519178-28-0, controls the biological activity of IP6K.
MilliporeSigma™ Calbiochem™ ODQ
A cell-permeable, potent and selective inhibitor of nitric oxide (NO)-sensitive guanylyl cyclase (IC50 = 20 nM).
MilliporeSigma™ Calbiochem™ PI 3-Kα Inhibitor IV
The PI 3-Kα Inhibitor IV, also referenced under CAS 1188890-32-5, controls the biological activity of PI 3-Kα. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ InSolution™ Purmorphamine
Purmorphamine is a cell-permeable purine compound that induces osteoblast differentiation in C3H10T1/2 multipotent mesenchymal progenitor cells.
MilliporeSigma™ Calbiochem™ Cathepsin D Substrate I
Useful as a substrate for the determination of cathepsin D activity.
MilliporeSigma™ Calbiochem™ Amyloid Precursor Protein β-Secretase Inhibitor
The Amyloid Precursor Protein β-Secretase Inhibitor controls the biological activity of Amyloid Precursor Protein β-Secretase. This small molecule/inhibitor is primarily used for Neuroscience applications.
MilliporeSigma™ Calbiochem™ NMDAR2C/2D Inhibitor, DQP-1105
The NMDAR2C/2D Inhibitor, DQP-1105 controls the biological activity of NMDAR2C/2D. This small molecule/inhibitor is primarily used for Neuroscience applications.