Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ Tankyrase1/2 Inhibitor IV, JW55
The Tankyrase1/2 Inhibitor IV, JW55 controls the biological activity of Tankyrase1/2. This small molecule/inhibitor is primarily used for Biochemicals applications.
MilliporeSigma™ Calbiochem™ Calpain Inhibitor IV
The Calpain Inhibitor IV controls the biological activity of Calpain. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
MilliporeSigma™ Calbiochem™ VEGFR Tyrosine Kinase Inhibitor VI, AAL-993
The VEGFR Tyrosine Kinse Inhibitor VI, ALL-993, also referenced under CAS 269390-77-4, controls the biological activity of VEGFR Tyrosine Kinase. This small molecule/inhibitor is primarily used for Cancer applications.
MilliporeSigma™ Calbiochem™ PD 98059
PD 98059, CAS 167869-21-8, is a cell-permeable, selective & reversible inhibitor of MAP Kinase Kinase (MEK). Inhibits MAP Kinase activation and subsequent phosphorylation of MAP Kinase substrates.
MilliporeSigma™ Calbiochem™ InSolution™ SRT1720, HCl
A 25 mM (10 mg/650 μl) sterile-filtered solution of SRT1720, HCl in DMSO.
MilliporeSigma™ Calbiochem™ FK-506, Streptomyces sp.
Immunosuppressant that blocks T cell proliferation in vitro by inhibiting the generation of several lymphokines, especially IL-2.
MilliporeSigma™ Calbiochem™ MAGL Inhibitor III, JZL184
The MAGL Inhibitor III, JZL184, also referenced under CAS 1101854-58-3, controls the biological activity of MAGL.
MilliporeSigma™ Calbiochem™ Furin Inhibitor I
Furin Inhibitor I, is a peptidyl chloromethylketone that binds to the catalytic site of furin and blocks its activity.
MilliporeSigma™ Calbiochem™ p300/CBP Inhibitor VI, L002
A cell-permeable phenylsulfonyloxyiminocyclohexadienone compound that acts as a potent, selective, and reversible inhibitor of p300 histone acetyl transferase (IC50
MilliporeSigma™ Calbiochem™ SIRT1 Activator II
The SIRT1 Activator II, also referenced under CAS 374922-43-7, modulates the biological activity of SIRT1. This small molecule/inhibitor is primarily used for Biochemicals applications.
MilliporeSigma™ Calbiochem™ Transglutaminase 2 Inhibitor, ZDON
A cell-permeable, peptide-based, irreversible inhibitor of transglutaminase 2 (TG2; IC50 = 150nM for recombinant TG2). Reacts with the active site cysteine of TG2.
MilliporeSigma™ Calbiochem™ MTEP Hydrochloride
A non-competitive, potent antagonist highly selective for mGlu5 receptors (IC50 =
MilliporeSigma™ Calbiochem™ Olomoucine
A purine derivative that acts as a potent, reversible and selective inhibitor of p34cdk1/cyclin B and related kinases.
MilliporeSigma™ Calbiochem™ E-4031
A potent and selective inhibitor of the rapid type of inactivating inward-rectifying K+ current (IK, IR) (IC50 = 10 nM).
MilliporeSigma™ Calbiochem™ Nimodipine
An L-type Ca2+ channel blocker.