Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ GPR43 (FFA2) Agonist
The GPR43 (FFA2) Agonist controls the biological activity of GPR43. This small molecule/inhibitor is primarily used for Biochemicals applications.
MilliporeSigma™ Calbiochem™ Collagenase Inhibitor I
The Collagenase Inhibitor I controls the biological activity of Collagenase. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
MilliporeSigma™ Calbiochem™ 3,4-Dichloroisocoumarin
A potent irreversible inhibitor of serine proteases
MilliporeSigma™ Calbiochem™ Histone Methyltransferase EZH2 Inhibitor, DZNep
Histone Methyltransferase EZH2 Inhibitor, DZNep, CAS 120964-45-6, is a cell-permeable inhibitor of EZH2-mediated trimethylation of K27 on histone H3.
MilliporeSigma™ Calbiochem™ Dantrolene, Sodium Salt
A cell-permeable blocker of intracellular calcium release from the sarcoplasmic reticulum that acts by binding to the ryanodine receptor.
MilliporeSigma™ Calbiochem™ Cyclophosphamide Monohydrate
A widely used anti-neoplastic agent that also displays immunosuppressant properties.
MilliporeSigma™ Calbiochem™ Sphingosine Kinase-2 Inhibitor, K145
A cell permeable, selective, sphingosine competitive inhibitor of spingosine Kinase -2 (IC50 = 4.3 μM).
MilliporeSigma™ Calbiochem™ InSolution™ Roscovitine
A potent and selective inhibitor of cyclin-dependent kinases (Cdks)
MilliporeSigma™ Calbiochem™ Pyruvate Kinase Activator
The Pyruvate Kinase Activator controls the biological activity of Pyruvate Kinase. This small molecule/inhibitor is primarily used for Activators/Inducers applications.
MilliporeSigma™ Calbiochem™ MICAL-2 Inhibitor II, CCG-203971
A cell-permeable, restricted form of CCG-1423 with enhanced potency (IC50 = 4.2 μM vs 16.6 μM for PC-3 cell migration), but reduced off-target toxicity.
MilliporeSigma™ Calbiochem™ bpV(phen)
A potent protein phosphotyrosine phosphatase inhibitor and insulin receptor kinase (IRK) activator.
MilliporeSigma™ Calbiochem™ Chk2 Inhibitor
The Chk2 Inhibitor, also referenced under CAS 724708-21-8, controls the biological activity of Chk2. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Swainsonine, Swainsona canescens
Reversible active-site inhibitor of lysosomal α-mannosidase.
MilliporeSigma™ Calbiochem™ EGFR Activator, NSC 228155
A nitro-benzoxadiazole compound that directly binds to the dimerization domain of sEGF receptor to generate stable dimers and allosterically activate the receptor.
MilliporeSigma™ Calbiochem™ Cathepsin L Inhibitor I
The Cathepsin L Inhibitor I, also referenced under CAS 108005-94-3, controls the biological activity of Cathepsin L. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.