Cycloheptathiophenes
Medchemexpress LLC Ocifisertib (fumarate) | 1616420-30-4 | 99.3% | 650.72 g/mol | C37H38N4O7 | 10MG
Ocifisertib fumarate is the fumarate salt of CFI-400945, an orally bioavailable small-molecule inhibitor of Polo-like kinase 4 (PLK4) for preclinical research. It is supplied as a powder for in vitro and in vivo studies and shows low-nanomolar potency against PLK4 and activity against several related kinases.
Medchemexpress LLC Formoterol fumarate | 43229-80-7 | >99.9% | C19H24N2O4 . 1/2C4H4O4 | 1 ML
Formoterol fumarate is a selective β2-adrenoceptor agonist, demonstrating similar β2-adrenoceptor selectivity to Salbutamol and Terbutaline. This compound is known for its ability to abolish the contraction induced by Acetylcholine in bronchioles. It is commonly utilized in research applications for conditions such as chronic obstructive pulmonary disease and bronchial asthma.
- Selective β2-adrenoceptor agonist
- Abolishes acetylcholine-induced contraction in bronchioles
- Used in research for chronic obstructive pulmonary disease
- Utilized in research for bronchial asthma
Medchemexpress LLC Bedaquiline fumarate | 845533-86-0 | 99.98% | 671.58 | 50 MG
Bedaquiline fumarate is an analytical standard and a diarylquinoline antibiotic that targets ATP synthase. It is effective for the treatment of Mycobacterium tuberculosis infections and is intended for research and analytical applications.
- Analytical standard grade
- Reference standard supplied assay
- Effective against Mycobacterium tuberculosis infections
- Commonly used in qualitative, quantitative, and methodological research experiments
- Suitable for HPLC, GC, and MS applications
Medchemexpress LLC Diethyl fumarate | 623-91-6 | 99.0% | 172.18 | 10 G
Diethyl fumarate is a decomposition product of Malathion 9 and a reactant in the Diels-Alder reaction. It is a reputed skin irritant and can cause non-immunologic contact urticaria on the skin. Diethyl fumarate and Curcumin hybridize to exert neuroprotective effects.
- Decomposition product of Malathion 9.
- Reactant in Diels-Alder reaction.
- Causes dose-dependent swelling of ears in guinea pigs.
- Curcumin hybrids show neuroprotective effects in C. elegans model of PD.
- For research use only.
Medchemexpress LLC Ocifisertib (fumarate) | 1616420-30-4 | 99.3% | 650.72 g/mol | C37H38N4O7 | 100MG
Ocifisertib (fumarate) is the fumarate salt form of a potent and selective ATP-competitive inhibitor of polo-like kinase 4 (PLK4) supplied for laboratory research. It is provided as a solid research reagent with molecular formula C37H38N4O7 and molecular weight 650.72 g/mol.
Medchemexpress LLC Ketotifen fumarate | 34580-14-8 | 99.9% | 25 MG
Ketotifen fumarate is an orally active second-generation noncompetitive histamine 1 (H1) receptor blocker and mast cell stabilizer. It can block 6-phosphogluconate dehydrogenase (PGD) in vitro. This compound also exhibits antiviral activity against SARS-CoV-2 and Influenza virus, making it useful in research for autoimmune encephalomyelitis (EAE) and the prevention of asthma attacks.
- Acts as an orally active second-generation noncompetitive histamine 1 (H1) receptor blocker
- Functions as a mast cell stabilizer
- Blocks 6-phosphogluconate dehydrogenase (PGD) in vitro
- Exhibits antiviral activity against SARS-CoV-2 and influenza virus
- Useful for research related to autoimmune encephalomyelitis (EAE)
- Applied in the prevention of asthma attacks research
Medchemexpress LLC Bedaquiline (fumarate) | 845533-86-0 | 99.99% | 671.58 | 25 MG
Bedaquiline (fumarate) is a diarylquinoline antibiotic that targets ATP synthase and is effective for the treatment of Mycobacterium tuberculosis infections. It inhibits the growth of TDR M. tuberculosis strains and shows high activity against Mycobacterium avium and moderate activity against NTM species. This product is for research use only.
- Targets ATP synthase
- Effective for treating Mycobacterium tuberculosis infections
- Inhibits growth of TDR M. tuberculosis strains
- High activity against Mycobacterium avium
- Moderate activity against NTM species
- For research use only