Oxazinanes
Medchemexpress LLC Pyrithioxin dihydrochloride | 10049-83-9 | 98.0% | 500 MG
Pyrithioxin (Pyritinol) dihydrochloride is the dihydrochloride salt of Pyrithioxin. Pyrithioxin (Pyritinol) is an orally active neurodynamic compound. Pyrithioxin can promote the metabolism of glucose and amino acids, increase carotid blood flow and improve cerebral blood flow. Pyrithioxin exhibits anti-inflammation, anti-tumor and neuroprotective effect. Pyrithioxin can be used for the researches of cancer, inflammation, immunology, metabolic and neurological disease such as cerebral infarct, epilepsy, fibrosarcomas and rheumatoid polyarthritis.
- Promotes metabolism of glucose and amino acids
- Increases carotid blood flow and improves cerebral blood flow
- Exhibits anti-inflammation effects
- Exhibits anti-tumor effects
- Provides neuroprotective effects
TARGETMOL CHEMICALS INC DROBULINE HYDROCHLORIDE 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Drobuline hydrochloride is an anti-arrhythmic agent with cardiac depressant activity. purity: 98%
TARGETMOL CHEMICALS INC CHK1-IN-4 HYDROCHLORIDE 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg and bulk. Please contact Fisher for quotes. CHK1-IN-4 hydrochloride is a potent inhibitor of checkpoint kinase 1 (chk1). CHK1-IN-4 hydrochloride potently inhibits chk1 phosphorylation in the tumor cells. CHK1-IN-4 hydrochloride has anti-tumor activity.
Medchemexpress LLC Clobenpropit dihydrobromide | 145231-35-2 | MFCD00467655 | 99.8% | 470.65 g/mol | C14H19Br2ClN4S | 50 MG
Clobenpropit dihydrobromide is a high-purity research chemical used as a potent histamine H3 receptor antagonist/inverse agonist and a partial H4 receptor agonist. Supplied as a white to off-white solid, it is intended for pharmacology and neuroscience studies to investigate histaminergic signaling and receptor pharmacology.
- High reported purity (99.76%).
- Molecular weight 470.65 g/mol; formula C14H19Br2ClN4S.
- White to off-white solid form suitable for in vitro and in vivo research.
- Recommended storage: 4°C sealed; in solvent -80°C up to 6 months.
- Potent nanomolar activity at histamine H3 and partial activity at H4; reported off-target binding to 5-HT3 and α2 adrenoceptors.
Medchemexpress LLC M-PEG12-Br | 1620461-89-3 | C25H51BrO12 | 250 MG
m-PEG12-Br is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs. It is for research use only and not sold to patients. PROTACs contain two different ligands connected by a linker; one is a ligand for an E3 ubiquitin ligase and the other is for the target protein. PROTACs exploit the intracellular ubiquitin-proteasome system to selectively degrade target proteins.
- Key component in the creation of PROTACs.
- Functions by connecting a ligand for an E3 ubiquitin ligase with a ligand for a target protein.
- Harnesses the intracellular ubiquitin-proteasome system for the selective degradation of target proteins.
eMolecules 957472-02-5 | (Z)-ETHYL 2-(PIPERIDIN-3-YLIDENE)ACETATE HCL | AstaTech | MFCD22573314 | 205.680 | C9H16ClNO2 | 96.000 | Cl.CCOC(=O)\C=C1\CCCNC1 | 1g | 290684257
(Z)-ETHYL 2-(PIPERIDIN-3-YLIDENE)ACETATE HCL | AstaTech | 957472-02-5 | MFCD22573314 | 205.680 | C9H16ClNO2 | 96.000 | Cl.CCOC(=O)\C=C1\CCCNC1 | 1g | 290684257
eMolecules 7778-42-9 | Sulfamoyl chloride | Oakwood Chemical | MFCD11519990 | 115.530 | ClH2NO2S | 95.000 | NS(Cl)(=O)=O | 250mg | 806975989
Sulfamoyl chloride | Oakwood Chemical | 7778-42-9 | MFCD11519990 | 115.530 | ClH2NO2S | 95.000 | NS(Cl)(=O)=O | 250mg | 806975989
eMolecules 121492-06-6 | N-Boc-N-methylethylenediamine | Ambeed | MFCD01317789 | 174.244 | C8H18N2O2 | 98.000 | CN(CCN)C(=O)OC(C)(C)C | 25g | 552722211
N-Boc-N-methylethylenediamine | Ambeed | 121492-06-6 | MFCD01317789 | 174.244 | C8H18N2O2 | 98.000 | CN(CCN)C(=O)OC(C)(C)C | 25g | 552722211
eMolecules 81893-75-6 | 4-(Methylamino)butanoic acid ethyl ester HCl | Acrotein ChemBio Inc. | MFCD17215565 | 181.660 | C7H16ClNO2 | 97.000 | Cl.CCOC(=O)CCCNC | 1g | 705837559
4-(Methylamino)butanoic acid ethyl ester HCl | Acrotein ChemBio Inc. | 81893-75-6 | MFCD17215565 | 181.660 | C7H16ClNO2 | 97.000 | Cl.CCOC(=O)CCCNC | 1g | 705837559
TARGETMOL CHEMICALS INC K145 HYDROCHLORIDE 50MG
Also available in 5 mg 10 mg 25 mg and bulk. Please contact Fisher for quotes. K145 hydrochloride is a selective sphk2 inhibitor with substrate competitiveness and oral activity with IC50 of 4.3 µM and Ki of 6.4 µM. K145 hydrochloride can induce apoptosis and has strong antitumor activity. purity: 99%
Cayman Chemical FR122047 hydrochloride
A selective COX-1 inhibitor (IC50 = 0.028 µM for the human enzyme); selective for COX-1 over COX-2 (IC50 = 65 µM); inhibits arachidonic acid, collagen, and ADP-induced platelet aggregation in human platelet-rich plasma (IC50 = 180-200 nM); unlike aspirin, it does not induce gastric damage at 100 mg/kg, p.o.; has an anti-inflammatory effect in a rat models of collagen-induced arthritis
TARGETMOL CHEMICALS INC CC-401 HYDROCHLORIDE 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. CC-401 Hydrochloride (CC401 HCl) is a second generation ATP-competitive anthrapyrazolone c-Jun N terminal kinase (JNK) inhibitor (Ki of 25 to 50 nM.)with potential antineoplastic activity. purity: 98%
TARGETMOL CHEMICALS INC KL-11743 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. KL-11743 specifically blocks glucose metabolism triggering an acute collapse in NADH pools and a striking accumulation of aspartate indicating a dramatic shift toward oxidative phosphorylation in the mitochondria. purity: 98%
Medchemexpress LLC Clobenpropit dihydrobromide | 145231-35-2 | MFCD00467655 | 99.8% | 470.65 g·mol⁻¹ | C14H19Br2ClN4S | 10 MG
Clobenpropit dihydrobromide is the dihydrobromide salt of clobenpropit, a histamine receptor ligand used for laboratory research. It acts as a potent histamine H3 receptor antagonist/inverse agonist and a partial H4 agonist, with reported additional binding to 5-HT3 and α2 adrenoceptors. The compound is supplied as a high-purity solid for receptor pharmacology and binding studies.
- High purity (99.76%).
- Molecular formula C14H19Br2ClN4S; molecular weight 470.65 g·mol⁻¹.
- CAS number 145231-35-2.
- Potent H3 antagonist/inverse agonist (pEC50 ~8.07).
- Suitable for receptor pharmacology and binding assays.
- Available in small research quantities (e.g., 10 MG).