Aminophenols
Medchemexpress LLC 3-pyridinecarboxylic acid, 1,2,5,6-tetrahydro-, hydrochloride | 6027-91-4 | MFCD00055191 | 99.9% | 163.60 g/mol | C6H10ClNO2 | 50 MG
Guvacine hydrochloride is the hydrochloride salt of guvacine, a pyridine alkaloid that inhibits GABA transporters. Supplied for research use to study GABA uptake and transporter pharmacology, it has reported activity across cloned human and rat GAT subtypes.
- Inhibits GABA transporter activity; reported IC50s include 14 μM (human GAT-1).
- High purity (≈99.9%) confirmed by COA.
- Molecular weight 163.60 g/mol; molecular formula C6H10ClNO2.
- Available in multiple pack sizes, including 50 mg, and solution formats in DMSO.
- Suitable for biochemical assays and transporter studies.
- Supplied with analytical documentation such as datasheet and COA.
Sigma Aldrich Fine Chemicals Biosciences Balsalazide Related Compound A United States Pharmacopeia (USP) Reference Standard | 1242567-07-2 (free acid) | 100MG
Balsalazide Related Compound A United States Pharmacopeia (USP) Reference Standard | Mol Wt: 330.2 | 1242567-07-2 (free acid) | 100MG
Selleck Chemical LLC 3-Hydroxybenzoic acid
3-Hydroxybenzoic acid (m-Hydroxybenzoic acid 3-Carboxyphenol m-Salicylic acid) is used as an intermediate in the synthesis of plasticisers resins pharmaceuticals etc
Medchemexpress LLC MRE-269-d7 | 1265295-20-2 | 99.6% | C25H22D7N3O3 | 1 MG
MRE-269-d7 is a deuterium-labeled form of MRE-269. It functions as an active metabolite of selexipag and acts as a selective IP receptor agonist. Stable heavy isotopes, such as deuterium, are incorporated into drug molecules primarily as tracers for quantitative analysis during drug development. Deuteration can also impact the pharmacokinetic and metabolic profiles of drugs.
- This compound can be used as a tracer.
- It can be used as an internal standard for quantitative analysis.
- It is an isotope-labeled compound.
- It is suitable for use in in vivo cell experiments.
- It is useful for therapeutic drug monitoring.
Medchemexpress LLC Melk-8a hydrochloride | 2096992-20-8 | 99.3% | 469.02 g·mol⁻¹ | C25H33ClN6O | 1 ML
MELK-8a hydrochloride is a small-molecule inhibitor of maternal embryonic leucine zipper kinase (MELK) with an in vitro IC50 of 2 nM. It is provided for research use in solution and solid formats and is used in biochemical and cellular studies to probe MELK-associated signaling pathways.
- Potent MELK inhibitor with an IC50 of 2 nM.
- Supplied as a 10 mM solution in DMSO (1 mL) and as solids (5-500 mg).
- High purity (≈99.3%) suitable for research applications.
- Molecular weight 469.02 g·mol⁻¹.
- CAS number 2096992-20-8 for unambiguous identification.
- For research use only; not for human or clinical use.
Medchemexpress LLC DI-82 | 1638148-50-1 | MFCD28386371 | 98.0% | 510.65 g·mol⁻¹ | C20H26N6O4S3 | 5 MG
DI-82 is a small-molecule inhibitor of deoxycytidine kinase (dCK) with reported biochemical potency and observed antitumor activity. It is supplied for research use in biochemical assays and preclinical studies as a powder form for laboratory workflows.
- Potent dCK inhibition: IC50app 27.8 nM; Kiapp 9.2 nM.
- High purity (98.0%) suitable for research applications.
- Soluble in DMSO at 120 mg/mL; ultrasonic assistance may be needed.
- Provided as a powder with recommended storage: -20°C for powder; -80°C for long-term storage in solvent.
- Intended for in vitro studies and preclinical antitumor research.
Medchemexpress LLC Gr 127935 hydrochloride | 148642-42-6 | MFCD08056244 | 99.4% | 534.05 | C29H32ClN5O3 | 10 MG
GR127935 hydrochloride is a potent, orally active antagonist of 5-HT1D and 5-HT1B serotonin receptors used in neurological and pharmacological research. Supplied as a white to off-white solid, it is characterized by high purity and documented solubility and storage recommendations for reliable experimental use.
- High purity suitable for research applications.
- Potent 5-HT1D and 5-HT1B receptor antagonism for receptor pharmacology studies.
- Supplied in small milligram quantities for in vitro and in vivo dosing.
- Soluble in DMSO; follow recommended handling and storage.
- Documentation includes datasheet, certificate of analysis, and safety data sheet for traceability.
Medchemexpress LLC Pirmenol hydrochloride | 61477-94-9 | MFCD01691662 | 98.8% | 374.95 g/mol | C22H31ClN2O | 10 MG
Pirmenol hydrochloride is the hydrochloride salt of pirmenol, an orally active research compound used to study cardiac ion channels and muscarinic acetylcholine receptor (mAChR) modulation. Supplied as a solid with batch-specific certificate of analysis documentation, this material is intended for laboratory research and screening applications where small, accurately dosed quantities are required.
- High chemical purity suitable for research use.
- Available in small milligram pack sizes for screening and assays.
- Supplied as a hydrochloride salt for improved handling and stability.
- Batch-specific certificate of analysis available for traceability.
- Appropriate for studies of ion channel function and muscarinic receptor activity.
Medchemexpress LLC HAIYPRH hydrochloride | 100.0% | 929.46 | 5 MG
HAIYPRH hydrochloride is a targeting ligand that specifically binds to the transferrin receptor (TfR). It can mediate the transport of nanocarriers across the blood-brain barrier.
- Can be conjugated to liposomes for ischemic stroke targeting treatment.
- Heptapeptide that can be used to target gliomas.
- Used as a ligand to target co-delivery systems to tumor cells expressing transferrin receptors.
- Modified co-delivery systems show higher efficiency in cellular uptake and gene expression in U87 MG cells.
- Modified co-delivery systems accumulate in tumors more efficiently in vivo.
Medchemexpress LLC 1-myristoyl-sn-glycero-3-phosphatidylcholine-d7 | 95.4% | 474.62 | 1 MG
LysoPC(14:0/0:0)-d7 is a deuterium labeled lysophospholipid (LyP). It is a monoglycerophospholipid where a phosphorylcholine moiety occupies a glycerol substitution site. This product exhibits a potent antispasmodic effect and is for research use only.
- Can be used as a tracer.
- Can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS.
Medchemexpress LLC HLCL-61 hydrochloride | 1158279-20-9 | MFCD09446681 | 99.9% | 380.91 g/mol | C23H25ClN2O | 1 ML
HLCL-61 hydrochloride is a small-molecule inhibitor of protein arginine methyltransferase 5 (PRMT5) supplied for research use. It is provided as concentrated DMSO stock solutions and as solid material for in vitro and in vivo studies; not for human or veterinary use.
- First-in-class PRMT5 inhibitor for research applications.
- Available as 10 mM stock solutions in DMSO and as solids in multiple sizes.
- High reported purity (approximately 99.9%).
- Soluble in DMSO (≈131 mM at 50 mg/mL) and poorly soluble in water.
- Storage: sealed at 4°C for solids; in solvent -80°C for long-term storage.
- Identifying information: CAS number 1158279-20-9; molecular weight ≈380.91 g/mol.
TARGETMOL CHEMICALS INC 4-Methylhistamine hydrochlorid
Also available in 1 mL, 1 mg, 2 mg, 10 mg, 25 mg, 50 mg, 100 mg, 500 mg and bulk. Please contact Fisher for quotes. 4-Methylhistamine hydrochloride has been shown to inhibit the activity of copper-dependent enzymes such as tyrosinase and dopamine beta-hydroxylase and has also been shown to modulate the expression of genes involved in cell cycle regulation and apoptosis. Purity 95%