Aminophenols
Medchemexpress LLC AZD9056 hydrochloride | 345303-91-5 | 98.2% | 455.46 | 50 MG
AZD9056 hydrochloride is a selective orally active inhibitor of P2X7, which plays a significant role in inflammation and pain-causing diseases. It is for research use only and not sold to patients.
- Selective orally active inhibitor of P2X7.
- Blocks P2X7 receptors with an IC50 of 11.2 nM in HEK-hP2X7 cell line.
- Exhibits high selectivity for the P2X7 receptor.
- Has an inhibitory effect (IC50=1-3 μM) in mouse microglia BV2 cells.
- Weakly inhibits BCRP-mediated transport of methotrexate (IC50=92 μM).
- Exerts pain-relieving and anti-inflammatory effects in vivo.
- Reverses upregulated expression of IL-1β, IL-6, TNF-α, MMP-13, SP, and PGE2 induced by MIA in cartilage tissues.
eMolecules 161265-03-8 | Xantphos | Ambeed | MFCD00233866 | 578.632 | C39H32OP2 | 98.000 | CC1(C)c2cccc(P(c3ccccc3)c3ccccc3)c2Oc2c(cccc12)P(c1ccccc1)c1ccccc1 | 25g | 552589291
Xantphos | Ambeed | 161265-03-8 | MFCD00233866 | 578.632 | C39H32OP2 | 98.000 | CC1(C)c2cccc(P(c3ccccc3)c3ccccc3)c2Oc2c(cccc12)P(c1ccccc1)c1ccccc1 | 25g | 552589291
Medchemexpress LLC Harmine hydrochloride | 343-27-1 | MFCD00078028 | 248.71 | 1 ML
Harmine hydrochloride, also known as Telepathine hydrochloride, is a natural DYRK inhibitor. It exhibits anticancer and anti-inflammatory activities, and has a high affinity for the 5-HT2A serotonin receptor. It is supplied as a solution in DMSO.
- Natural DYRK inhibitor
- Exhibits anticancer and anti-inflammatory activities
- High affinity for 5-HT2A serotonin receptor
- Supplied in solution for convenience
Medchemexpress LLC Irigenin | 548-76-5 | MFCD00597047 | 99.8% | 360.31 g/mol | C18H16O8 | 10 MG
Irigenin is an isoflavone research compound used to inhibit Extra Domain A (EDA)-integrin interactions and to study integrin-mediated signaling and apoptosis in vitro. It is supplied as a solid powder and as DMSO solutions for assay preparation.
- Inhibits EDA-integrin interactions and is used in integrin and apoptosis research.
- High purity (99.84%) suitable for research applications.
- Molecular weight 360.31 g/mol; chemical formula C18H16O8.
- CAS number 548-76-5 for unambiguous identification.
- Available as solid powder and 10 mM solutions in DMSO for assay use.
- Available in small research pack sizes including 10 MG.
Medchemexpress LLC YIL781 hydrochloride | 1640226-17-0 | 99.5% | 445.96 g/mol | C24H29ClFN3O2 | 5 MG
YIL781 hydrochloride is the hydrochloride salt of a potent, orally active ghrelin receptor (GHSR) antagonist used in preclinical research to study ghrelin signaling, metabolic regulation, and insulin secretion. The compound is provided with solubility guidance and storage recommendations for reliable use in experimental workflows.
- Potent ghrelin receptor (GHSR) antagonist suitable for pharmacological studies.
- Usable in vitro and in vivo applications.
- High purity (~99.5%) for reliable experimental results.
- Soluble in DMSO; formulation guidance provided for aqueous preparations.
- Stable when stored sealed at -20°C; solvent stability recommendations available.
- Available in small research pack sizes for early-stage studies.
Medchemexpress LLC Cyclohexanecarboxylic acid, 1-phenyl-, 2-(4-morpholinyl)ethyl ester, hydrochloride (1:1) | 75136-54-8 | 99.8% | 353.88 | 1 ML
PRE-084 hydrochloride is a highly selective σ1 receptor (S1R) agonist, with an IC50 of 44 nM. It exhibits good neuroprotective effects, can improve motor function and motor neuron survival in mice, and can ameliorate myocardial ischemia-reperfusion injury in rats by activating the Akt-eNOS pathway.
- Highly selective σ1 receptor (S1R) agonist (IC50 of 44 nM).
- Exhibits neuroprotective effects.
- Improves motor function and motor neuron survival in mice.
- Ameliorates myocardial ischemia-reperfusion injury in rats by activating the Akt-eNOS pathway.
Medchemexpress LLC Histidyl-proline hydrochloride | 2415727-78-3 | 99.8% | 288.73 g·mol⁻¹ | C11H17ClN4O3 | 5 MG
His-Pro hydrochloride (histidyl-proline hydrochloride) is a research-grade dipeptide composed of histidyl and proline supplied as the hydrochloride salt. Offered as a white to off-white powder, it is intended for analytical and biochemical applications including peptide research and assay development.
- High purity (~99.8%) suitable for analytical work.
- Molecular weight 288.73 g·mol⁻¹.
- Chemical formula C11H17ClN4O3.
- Available in small, milligram-scale quantities for research use.
- Solid powder form with recommended refrigerated storage to preserve stability.
eMolecules 103-90-2 | Acetaminophen | Combi-Blocks | MFCD00002328 | 151.165 | C8H9NO2 | 98.000 | CC(=O)Nc1ccc(O)cc1 | 5g | 335345644
Acetaminophen | Combi-Blocks | 103-90-2 | MFCD00002328 | 151.165 | C8H9NO2 | 98.000 | CC(=O)Nc1ccc(O)cc1 | 5g | 335345644
Medchemexpress LLC CGP71683 hydrochloride | 192322-50-2 | MFCD07783999 | 99.4% | 512.07 g/mol | C26H30ClN5O2S | 50 MG
CGP71683 hydrochloride is a selective, non-peptide neuropeptide Y (NPY) Y5 receptor antagonist used for in vitro pharmacology and receptor signaling studies. The compound is supplied as a white solid and as a 10 mM solution in DMSO and is reported with high purity for research applications.
- Selective NPY Y5 receptor antagonist with low nanomolar affinity.
- Reported high purity suitable for research use.
- Available as a solid and as a 10 mM solution in DMSO for assay convenience.
- Molecular weight 512.07 g/mol aiding stoichiometric calculations.
- CAS registry number 192322-50-2 for unambiguous identification.
- Intended for biochemical and pharmacological studies in vitro.
eMolecules 202475-60-3 | JANEX-1 | AstaTech | MFCD01862614 | 297.314 | C16H15N3O3 | 95.000 | COc1cc2ncnc(Nc3ccc(O)cc3)c2cc1OC | 1g | 290663216
JANEX-1 | AstaTech | 202475-60-3 | MFCD01862614 | 297.314 | C16H15N3O3 | 95.000 | COc1cc2ncnc(Nc3ccc(O)cc3)c2cc1OC | 1g | 290663216
Medchemexpress LLC R 59-022 hydrochlori 10mg | 93076-98-3 | 10MG
R 59-022 (DKGI-I) hydrochloride is a DGK inhibitor (IC50 2 8 M) R 59-022 hydrochloride inhibits the phosphorylation of OAG to OAPA R 59-022 hydrochloride is a 5-HT Receptor antagonist and activates protein kinase C (PKC) R 59-022 hydrochloride potentiates thrombin-induced diacylglycerol production in platelets and inhibits phosphatidic acid production in neutrophils[1 [2 [3 [4