Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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2,581
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2,581
Tocris Bioscience™ AY 9944 dihydrochloride
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 366-93-8 Molecular Formula: C22H30Cl4N2
| CAS | 366-93-8 |
|---|---|
| Molecular Formula | C22H30Cl4N2 |
2,582
Tocris Bioscience™ L-Ascorbic acid
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CAS: 50-81-7 Molecular Formula: C6H8O6
| CAS | 50-81-7 |
|---|---|
| Molecular Formula | C6H8O6 |
2,583
Tocris Bioscience™ VU 0071063
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Selective activator of SUR1 Kir6.2 channels
| Target | Inward Rectifier Potassium Channel Activators |
|---|---|
| CAS | 333415-38-6 |
| Purity | 0.98 |
| Chemical Name or Material | 7-[[4-(1,1-Dimethylethyl)phenyl]methyl]-3,7-dihydro-1,3-dimethyl-1 H-purine-2,6-dione |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C18H22N4O2 |
2,584
Tocris Bioscience™ ASP 3026
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Potent anaplastic lymphoma kinase (ALK) inhibitor; also potent ACK inhibitor
| Target | ALK Inhibitors |
|---|---|
| CAS | 1097917-15-1 |
| Purity | >99% |
| Chemical Name or Material | N2-[2-Methoxy-4-[4-(4-methyl-1-piperazinyl)-1-piperidinyl]phenyl]-N4-[2-[(1-methylethyl)sulfonyl]phenyl]-1,3,5-triazine-2,4-diamine |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C29H40N8O3S |
| Formula Weight | 580.74 |
2,585
Tocris Bioscience™ Docetaxel
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CAS: 114977-28-5 Molecular Formula: C43H53NO14
| CAS | 114977-28-5 |
|---|---|
| Molecular Formula | C43H53NO14 |
2,586
Tocris Bioscience™ ML 299
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Potent inhibitor of PLD1 and PLD2; CNS penetrant
2,587
Tocris Bioscience™ DBM 1285 dihydrochloride
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p38 MAPK inhibitor; anti-inflammatory
| Inhibitors | DBM 1285 dihydrochloride |
|---|---|
| Product Type | DBM 1285 dihydrochloride |
| Molecular Weight (g/mol) | 468.42 |
| Purity | >98% |
2,588
Tocris Bioscience™ AZD 5363
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent pan-AKT inhibitor
| Product Type | Inhibitor |
|---|---|
| Purity | 98% |
| Recommended Storage | Store at -20°C |
| Synonym | Capivasertib |
| Molecular Formula | C21H25ClN6O2 |
| Formula Weight | 428.92 |
2,589
Tocris Bioscience™ LAP
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Photocrosslinker for hydrogels
2,590
Tocris Bioscience™ MTK 458
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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PINK1 activator
| Target | PINK1 |
|---|---|
| CAS | 2499962-58-0 |
| Purity | 0.98 |
| Chemical Name or Material | N-[(1R)-1,2,3,4-Tetrahydro-1-naphthalenyl]-6-(trifluoromethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C17H15F3N4 |
2,591
Tocris Bioscience™ BAY 9835
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Potent ADAMTS7 and ADAMTS12 inhibitor
| Target | Synthetic Metalloprotease Inhibitors |
|---|---|
| Recommended Storage | Store at -20°C |
2,592
Tocris Bioscience™ PNU 142633
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CAS: 187665-65-2 Molecular Formula: C24H30N4O3
| CAS | 187665-65-2 |
|---|---|
| Molecular Formula | C24H30N4O3 |
2,593
Tocris Bioscience™ (+)-Igmesine hydrochloride
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Selective sigma1 ligand; antidepressant
| CAS | 130152-35-1 |
|---|---|
| Solubility | Soluble to 50mM in DMSO |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C23H29N.HCl |
| Formula Weight | Observed MW: 355.94 |
| Assay Percent Range | >98% |
2,594
Tocris Bioscience™ TR 14035
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Potent integrin α4β7 and α4β1 (VLA-4) antagonist
| Product Type | Antagonist |
|---|---|
| Purity | 98% |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C24H21Cl2NO5 |
| Formula Weight | 474.33 |
2,595
Tocris Bioscience™ Rosiglitazone
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Potent and selective PPARγ agonist; antidiabetic agent
| Target | PPAR gamma Receptor Agonists |
|---|---|
| CAS | 122320-73-4 |
| Purity | 98% |
| Chemical Name or Material | 5-[[4-[2-(Methyl-2-pyridinylamino)ethoxy]phenyl]methyl]-2,4-thiazolidinedione |
| Recommended Storage | Store at 4°C |
| Synonym | BRL 49653 |
| Molecular Formula | C18H19N3O3S |
| Formula Weight | 357.43 |