Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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2,881
Tocris Bioscience™ AZD 7648
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Potent and selective DNA-PK inhibitor
| Target | DNA-dependent Protein Kinase Inhibitors |
|---|---|
| CAS | 2230820-11-6 |
| Chemical Name or Material | 7,9-Dihydro-7-methyl-2-[(7-methyl[1,2,4]triazolo[1,5-a]pyridin-6-yl)amino]-9-(tetrahydro-2H-pyran-4-yl)-8H-purin-8-one |
| Recommended Storage | Store the unopened product at -20 to -70 °C. Use a manual defrost freezer and avoid repeated freeze-thaw cycles. Do not use past expiration date. |
| Molecular Formula | C18H20N8O2 |
2,882
Tocris Bioscience™ GSK 2193874
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and selective TRPV4 antagonist; orally active
| CAS | 1336960-13-4 |
|---|---|
| Chemical Name or Material | 3-([1,4'-Bipiperidin]-1'-ylmethyl)-7-bromo-N-(1-phenylcyclopropyl)-2-[3-(trifluoromethyl)phenyl]-4-quinolinecarboxamide |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C37H38BrF3N4O |
| Formula Weight | Observed MW: 691.62 |
| Assay Percent Range | >98% |
2,883
Tocris Bioscience™ AMZ 30
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Potent, selective and irreversible protein phosphatase methylesterase-1 (PME-1) inhibitor
| Target | Hydrolase Inhibitors |
|---|---|
| CAS | 1313613-09-0 |
| Purity | 0.98 |
| Chemical Name or Material | (2 E)-2-[(4-Fluorophenyl)sulfonyl]-3-[1-[(3-nitrophenyl)sulfonyl]-1 H-pyrrol-2-yl]-2-propenenitrile |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C19H12FN3O6S2 |
2,884
Tocris Bioscience™ Asunaprevir
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Potent hepatitis C virus (HCV) NS3 protease inihibitor
| Target | CRISPR Reagents |
|---|---|
| CAS | 630420-16-5 |
| Purity | 0.98 |
| Chemical Name or Material | 1-[[N-tert-Butoxycarbonyl-L-tert-leucyl-trans-4-[(7-chloro-4-methoxyisoquinolin-1-yl)oxy]-L-prolyl]amino]-N-(cyclopropylsulfonyl)-(1 R,2 S)-2-vinylcyclopropane-1-carboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C35H46ClN5O9S |
2,885
Tocris Bioscience™ CL 316243 disodium salt
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CAS: 151126-84-0 Molecular Formula: C20H18ClNNaO7-
| CAS | 151126-84-0 |
|---|---|
| Molecular Formula | C20H18ClNNaO7- |
2,886
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Tocris Bioscience™ FTY 720
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Tocris Bioscience™ FTY 720
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent S1P receptor agonist; also immunosuppressant
| Target | Sphingosine-1-phosphate Receptor |
|---|---|
| CAS | 162359-56-0 |
| Product Type | Agonist |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C19H33NO2.HCl |
| Formula Weight | 343.93g/mol |
2,887
Tocris Bioscience™ (±)-J 113397
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 217461-40-0 Molecular Formula: C24H37N3O2
| CAS | 217461-40-0 |
|---|---|
| Molecular Formula | C24H37N3O2 |
2,888
Tocris Bioscience™ AS2717638
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Selective, brain penetrant LPA5 antagonist
2,889
Tocris Bioscience™ 2-BFI hydrochloride
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CAS: 89196-95-2 Molecular Formula: C11H11ClN2O
| CAS | 89196-95-2 |
|---|---|
| Molecular Formula | C11H11ClN2O |
2,890
Tocris Bioscience™ PJ 34 hydrochloride
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CAS: 344458-15-7 Molecular Formula: C17H18ClN3O2
| CAS | 344458-15-7 |
|---|---|
| Molecular Formula | C17H18ClN3O2 |
2,891
Tocris Bioscience™ TAK 21d
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Potent FAAH inhibitor
| Target | Fatty Acid Amide Hydrolase (FAAH) Inhibitors |
|---|---|
| CAS | 1143578-94-2 |
| Purity | >98% |
| Chemical Name or Material | 4-[4-(3,4-Difluorophenyl)-2-pyrimidinyl]-N-3-pyridazinyl-1-piperazinecarboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C19H17F2N7O |
| Formula Weight | 397.38 |
2,892
Tocris Bioscience™ CGP 36216 hydrochloride
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GABAB antagonist; displays activity at presynaptic receptors
| Inhibitors | CGP 36216 hydrochloride |
|---|---|
| CAS | 1781834-71-6 |
| Product Type | CGP 36216 hydrochloride |
| Molecular Weight (g/mol) | 187.6 |
| Purity | >99% |
2,893
Tocris Bioscience™ SR 10067
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Selective Rev-Erbα/β agonist; anxiolytic
| CAS | 1380548-02-6 |
|---|---|
| Chemical Name or Material | [3-[[4-(1,1-Dimethylethoxy)phenoxy]methyl]-3,4-dihydro-2(1H)-isoquinolinyl]-1-naphthalenylmethanone |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C31H31NO3 |
| Formula Weight | Observed MW: 465.58 |
| Assay Percent Range | >98% |
2,894
Tocris Bioscience™ SR 27897
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Potent and selective CCK1 antagonist
| Inhibitors | SR 27897 |
|---|---|
| Product Type | SR 27897 |
| Molecular Weight (g/mol) | 411.86 |
| Purity | >99% |
2,895
Tocris Bioscience™ WM 8014
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Potent and selective KAT6A and KAT6B inhibitor