Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ Methyl Arachidonyl Fluorophosphonate
A selective, active site-directed, irreversible inhibitor of both calcium-dependent and calcium-independent cytosolic (85 kDa) phospholipase A2 (PLA2) but not of secretory PLA2.
MilliporeSigma™ Calbiochem™ InSolution™ Ratjadone A, Synthetic
A cell-permeable polyketide that displays potent antitumor properties in eukaryotes.
MilliporeSigma™ Calbiochem™ Smac-N7 Peptide
A peptide that contains the N-terminal seven residues of Smac (Second Mitochondria-derived Activator of Caspases, also known as DIABLO) and promotes procaspase-3 activation at around 10μM.
MilliporeSigma™ Calbiochem™ SB 202474
A negative control for SB202190 and SB203580 in p38 MAP kinase inhibition studies.
MilliporeSigma™ Calbiochem™ MELK Inhibitor, OTSSP167
A cell permeable, orally bioavailable 1, 5-naphthyridine based compound that acts as a highly potent and specific inhibitor of maternal embryonic leucine zipper kinase (MELK; IC50 = 410)
MilliporeSigma™ Calbiochem™ BPDQ
A cell-permeable, reversible, ATP-competitive, potent and specific inhibitor of the tyrosine kinase activity of the epidermal growth factor receptor (EGFR; IC50 = 120 pM).
MilliporeSigma™ Calbiochem™ L-CCG-I
A potent agonist for group II metabotropic glutamate receptors (EC50
MilliporeSigma™ Calbiochem™ NG-Monomethyl-L-arginine, Monoacetate Salt
Cell permeable. L-Arginine analog that acts as a competitive inhibitor of all three isoforms of NOS.
MilliporeSigma™ Calbiochem™ 5-BDBD
A highly potent antagonist of purinergic P2X4 recep
Novus Biologicals™ Staurosporine Inhibitor
Low molecular weight, organic compound that may help regulate biological process.
Novus Biologicals™ Actinomycin D Inhibitor
Low molecular weight, organic compound that may help regulate biological process.
Novus Biologicals™ Z-DEVD-FMK Inhibitor
Low molecular weight, organic compound that may help regulate biological process.
MilliporeSigma™ Calbiochem™ EGFR Inhibitor II, BIBX1382
The EGFR Inhibitor II, BIBX1382, also referenced under CAS 196612-93-8, controls the biological activity of EGFR. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
Novus Biologicals™ Z-VAD-FMK Inhibitor
Low molecular weight, organic compound that may help regulate biological process.
MilliporeSigma™ Calbiochem™ Elastase Inhibitor I
The Elastase Inhibitor I controls the biological activity of Elastase. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.