Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ Akt Inhibitor XII, Isozyme-Selective, Akti-2
The Akt Inhibitor XII, Isozyme-Selective, Akti-2 controls the biological activity of Akt. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ MK2a Inhibitor
The MK2a Inhibitor, also referenced under CAS 41179-33-3, controls the biological activity of MK2a. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Cyclophilin A Inhibitor
The Cyclophilin A Inhibitor, also referenced under CAS 1186372-20-2, controls the biological activity of Cyclophilin A. This small molecule/inhibitor is primarily used for Inflammation/Immunology applications.
MilliporeSigma™ Calbiochem™ HIF-1 Inhibitor
The HIF-1 Inhibitor, also referenced under CAS 934593-90-5, controls the biological activity of HIF-1.
MilliporeSigma™ Calbiochem™ Akt Inhibitor X
The Akt Inhibitor X, also referenced under CAS 925681-41-0, controls the biological activity of Akt. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ MMP Substrate III, Fluorogenic
A specific fluorogenic resonance energy transfer (FRET) peptide substrate with an MMP cleavable Gly-Leu bond and EDANS/Dabcyl as fluorophore/quencher combination.
MilliporeSigma™ Calbiochem™ SNAPtide™ Botulinum Toxin A Substrate, Fluorogenic
SNAPtide™ Botulinum Toxin A Substrate, Fluorogenic, is a synthetic peptide that acts as a FRET substrate with the fluorophore o-aminobenzoic acid and the acceptor chromophore 2,4-dinitrophenol (DNP).
MilliporeSigma™ Calbiochem™ PPACK II, Trifluoroacetate Salt
Potent and specific irreversible inhibitor of plasma and glandular kallikreins.
MilliporeSigma™ Calbiochem™ Phenylmethylsulfonyl Fluoride
Phenylmethylsulfonyl Fluoride, CAS 329-98-6, is an irreversible inhibitor of serine proteases. It causes sulfonylation of the active-site serine residues.
MilliporeSigma™ Calbiochem™ AEBSF, HCl ≥99% by HPLC
Specific irreversible inhibitor of serine proteases
MilliporeSigma™ Calbiochem™ Picrotoxin, Anamirta cocculin
A potent antagonist of GABA receptors (IC50 = 240 nM) at synapses in the central nervous system.
MilliporeSigma™ Calbiochem™ Ro-20-1724
A cell-permeable, selective inhibitor of cAMP-specific phosphodiesterase (PDE IV; IC50 = 2 μM).
MilliporeSigma™ Calbiochem™ QX-314
A quaternary lidocaine derivative, permanently charged, and lipophobic.
MilliporeSigma™ Calbiochem™ PTP1B Inhibitor
PTP1B Inhibitor, CAS 765317-72-4, is a cell-permeable, selective, reversible and non-competitive allosteric inhibitor of PTP1B (IC50 = 4 μM and 8 μM for PTP1B403 and PTP1B298, respectively).
MilliporeSigma™ Calbiochem™ Quercetin, Dihydrate
A cell-permeable and reversible inhibitor of PIM1 kinase (IC50 = 43nM), PI 3-K (IC50 = 3.8μM) and phospholipase A2