Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ CFTR-F508del Corrector II, Corr-4a
A cell-permeable bisaminomethylbithiazole compound that is reported to rescue/correct the folding defect of CFTR δF508 mutant via direct interaction.
MilliporeSigma™ Calbiochem™ InSolution™ CFTR Inhibitor II, GlyH-101
A cell-permeable glycinyl hydrazone compound that acts as a potent, selective and reversible open-channel blocker of CFTR with intermediate speed (<1 min; 95% inhibition at 50μM; Ki
MilliporeSigma™ Calbiochem™ BMP Inhibitor II, DMH1
The BMP Inhibitor II, DMH1, also referenced under CAS 1206711-16-1, controls the biological activity of BMP. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Bryostatin 1
A macrocyclic lactone with antitumor properties.
MilliporeSigma™ Calbiochem™ BTS
A potent inhibitor of Ca2+-stimulated myosin S1 ATPase (IC50 = ≈5 μM) and reversibly blocks the gliding motility.
MilliporeSigma™ Calbiochem™ Caffeine
Trimethylated xanthine that acts as a potent central nervous system stimulant.
MilliporeSigma™ Calbiochem™ E-Cadherin Upregulator, ResEcad
A cell-permeable isoxazolocarboxamide compound that enhances the E-cadherin protein level in lung squamous cell carcinoma H520 and colorectal adenocarcinoma SW620 cells.
MilliporeSigma™ Calbiochem™ GSK-3β Inhibitor XI
The GSK-3β Inhibitor XI, also referenced under CAS 626604-39-5, controls the biological activity of GSK-3β. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ Pre-mRNA Splicing Inhibitor, Isoginkgetin
The Pre-mRNA Splicing Inhibitor, Isoginkgetin, also referenced under CAS 548-19-6, blocks the spliceosome-meidated splicing process.
MilliporeSigma™ Calbiochem™ JNK Inhibitor II
JNK Inhibitor II. SP600125, CAS 129-56-6, is a potent, cell-permeable, selective, and ATP competitive inhibitor of c-Jun N-terminal kinase (JNK; IC50 = 40 nM for JNK-1 & JNK-2 & 90 nM for JNK-3).
MilliporeSigma™ Calbiochem™ InSolution™ JNK Inhibitor II
The InSolution™ JNK Inhibitor II, also referenced under CAS 129-56-6, controls the biological activity of JNK. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
MilliporeSigma™ Calbiochem™ InSolution™ Jasplakinolide, Jaspis johnstoni
InSolution™ Jasplakinolide, Jaspis johnstoni, CAS 102396-24-7, is a 1mm solution of Jasplakinolide, Jaspis johnstoni in DMSO. Acts as a potent inducer of actin polymerization and stabilization.
MilliporeSigma™ Calbiochem™ K-252a, Nocardiopsis sp.
A cell-permeable, reversible, and ATP-competitive inhibitor against multiple protein kinases.
MilliporeSigma™ Calbiochem™ JNK Inhibitor XIII
The JNK Inhibitor XIII, also referenced under CAS 40045-50-9, controls the biological activity of JNK. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.