Hydrobromides
TARGETMOL CHEMICALS INC TAZEMETOSTAT HYDROBROMID 100MG
Also available in 2 mg 5 mg 10 mg 50 mg 200 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Tazemetostat hydrobromide (E-7438 hydrobromide) is a potent and selective EZH2 inhibitor. Tazemetostat hydrobromide inhibits the activity of human polycomb repressive complex 2 (PRC2)-containing wild-type EZH2 (Ki 2.5 nM). Tazemetostat hydrobromide also inhibits EZH1 (IC50 392 nM). purity: 99%
TARGETMOL CHEMICALS INC PIFITHRIN-BETA HYDROBROM 25MG
Also available in 2 mg 5 mg 10 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Pifithrin-(beta) hydrobromide (Cyclic PFT-(alpha)) is an inhibitor of p53; reversibly blocks p53-dependent transcriptional activation and apoptosis. Protects against neuronal death in models of stroke and neurodegenerative disorders. Active in vivo; protects mice from the side-effects of Y therapy associated with p53 induction. Supresses self-renewal of embryonic stem cells. Also aryl hydrocarbon receptor (AHR) agonist causes upregulation of AHR target gene CYP1A1 (EC50 = 1.1 uM). purity: 99%
Apexbio Technology LLC Arecoline hydrobromide 300-08-3 10mM (in 1mL DMSO)
Arecoline hydrobromide (CAS 300-08-3) is a nicotinic alkaloid that acts as a partial agonist at muscarinic acetylcholine receptors M1 M4 In electrophysiological studies it significantly inhibits the hERG potassium channel current with an IC50 of 9 55 mol/L The compound s inhibitory effect on IhERG displays concentration time and voltage dependency with blockade intensity influenced by stimulation frequency Subcutaneous administration in mice yields an LD50 of 100 mg/kg Arecoline hydrobromide is utilized in research on cardiac electrophysiology and muscarinic receptor pharmacology particularly for investigating frequency- and state-dependent modulation of cardiac ion channels
Medchemexpress LLC Amthamine dihydrobromide | 142457-00-9 | MFCD00673891 | 99.6% | 319.07 g·mol⁻¹ | C6H13Br2N3S | 25 MG
Amthamine dihydrobromide is the dihydrobromide salt of amthamine, a histamine receptor agonist active at H1-H4 receptors. It is supplied as a solid and in ready-to-use DMSO solution formats for pharmacological research, and includes storage recommendations for both solids and stock solutions.
Medchemexpress LLC Amthamine dihydrobromide | 142457-00-9 | MFCD00673891 | 99.6% | 319.07 g/mol | C6H13Br2N3S | 50 MG
Amthamine dihydrobromide is a research-grade histamine receptor agonist provided as the dihydrobromide salt. It is used in pharmacology and toxicology research to study histamine receptor activation and downstream physiological effects in vitro and in vivo.
- Selective histamine H2 receptor agonist.
- High chemical purity suitable for research applications.
- Available as a solid for flexible dosing and formulation.
- Includes molecular and CAS identifiers for unambiguous compound identification.
Medchemexpress LLC Pyrithiamine hydrobromide | 534-64-5 | 96.6% | 10MG
Pyrithiamine hydrobromide | 534-64-5 | 96.6% | 10MG
TARGETMOL CHEMICALS INC Teneligliptin hydrobromide
Also available in 5 mg, 10 mg, 25 mg, 100 mg, 200 mg, 500 mg and bulk. Please contact Fisher for quotes. Teneligliptin hydrobromide (MP-513 (hydrobromide)) is a novel, potent, and long-lasting dipeptidyl peptidase-4 inhibitor; competitively inhibited human plasma, rat plasma, and human recombinant DPP-4 in vitro, with IC50 values of approximately 1 nM. Purity 100%