Cycloheptathiophenes
TARGETMOL CHEMICALS INC KT-362 FUMARATE 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. KT-362 fumarate is a novel compound that acts as an antagonist of calcium channels potassium channels and sodium channels.KT-362 fumarate causes vasodilation by affecting intracellular calcium mobilization in atrial muscle cells.KT-362 fumarate has a relaxing effect on femoral and basilar artery strips in rabbits. purity: 99%
Apexbio Technology LLC Ibutilide Fumarate 122647-32-9 100mg
Ibutilide Fumarate (CAS 122647-32-9) is a small molecule classified as a Class III antiarrhythmic agent It acts primarily by enhancing slow inward sodium currents and delaying repolarization through inhibition of the rapid component of the cardiac delayed rectifier potassium current (IKr) resulting in prolongation of the cardiac action potential Ibutilide is utilized in research to investigate pharmacological cardioversion of atrial arrhythmias specifically studying the acute conversion of atrial fibrillation and atrial flutter to normal sinus rhythm Its properties make it valuable for exploring the mechanisms of antiarrhythmic therapy and cardiac electrophysiology
Medchemexpress LLC Monomethyl fumarate-d2 | 253122-44-0 | MFCD00063174 | 98.2% | 132.11 | C5H4D2O4 | 1 MG
Monomethyl fumarate-d2 is the deuterium-labeled form of monomethyl fumarate, provided as a high-purity research chemical and isotopically labeled standard for metabolic, pharmacological, and analytical studies.
- Deuterium-labeled analog for isotope tracing and mass spectrometry.
- High purity suitable for research applications.
- Supplied in milligram quantities for small-scale experiments.
- Useful as a metabolic standard and mechanistic probe.
Medchemexpress LLC Ocifisertib fumarate | 1616420-30-4 | >98.0% | 650.7 g/mol | C37H38N4O7 | 50MG
Ocifisertib fumarate is the fumarate salt of CFI-400945, a potent, selective, and orally bioavailable inhibitor of polo-like kinase 4 (PLK4) supplied for research use in biochemical and cellular studies of PLK4-related pathways and antineoplastic activity.
- Fumarate salt form of the PLK4 inhibitor.
- Potent biochemical activity: PLK4 Ki = 0.26 nM; PLK4 IC50 = 2.8 nM.
- Molecular formula C37H38N4O7 and molecular weight 650.7 g/mol.
- High purity (>98.0% by HPLC) suitable for research applications.
- Supplied in small research pack sizes, including 50 mg.
Medchemexpress LLC Ocifisertib (fumarate) | 1616420-30-4 | 99.3% | 650.72 g/mol | C37H38N4O7 | 10MG
Ocifisertib fumarate is the fumarate salt of CFI-400945, an orally bioavailable small-molecule inhibitor of Polo-like kinase 4 (PLK4) for preclinical research. It is supplied as a powder for in vitro and in vivo studies and shows low-nanomolar potency against PLK4 and activity against several related kinases.
Medchemexpress LLC Zamifenacin fumarate | 127308-98-9 | 99.0% | 531.60 g/mol | C31H33NO7 | 1 ML
Zamifenacin fumarate is a gut-selective muscarinic M3 receptor antagonist provided for research use. It reduces colonic motility and is commonly used in pharmacology studies of muscarinic receptor function. The compound is available as a solid or as pre-made DMSO solution (typical 10 mM, 1 mL), with reported purity around 99.0% and molecular weight 531.60 g/mol.
Medchemexpress LLC Iron(II) fumarate (Ferrous fumarate) | 141-01-5 | 95.1% | 1 G
Iron (II) fumarate is an orally effective active dietary supplement. It can alleviate metabolic damage and damage to silkworms caused by cypermethrin and can be used for research on iron deficiency anemia.
- In vitro: Can restore metabolic pathway disruption and enhance cell viability in BmN cells treated with cypermethrin.
- In vivo: Alleviates damage caused by cypermethrin in silkworms.
- In vivo: Induces oxidative stress in the liver and colon of rats.
- In vivo: Alters intestinal morphology and microbiota in Yellow River carp, increasing diversity and richness.
Medchemexpress LLC Ensitrelvir fumarate | 2757470-18-9 | 99.99% | C26H21ClF3N9O6 | 25 MG
Ensitrelvir fumarate is an orally active, non-covalent, and non-peptidic SARS-CoV-2 3CL protease inhibitor. It demonstrates significant inhibitory activity against various SARS-CoV-2 variants and has shown to inhibit intrapulmonary replication of SARS-CoV-2 in mice.
- First orally active non-covalent, non-peptidic SARS-CoV-2 3CL protease inhibitor
- Shows EC50 values of approximately 0.4 μM for wild-type and Alpha, Beta, Gamma, and Delta SARS-CoV-2 variants
- Inhibits intrapulmonary replication of SARS-CoV-2 in mice
- For research use only
Medchemexpress LLC 2-butenedioic acid (2E)-, 1-ethyl ester | 2459-05-4 | MFCD00002699 | 99.6% | 144.13 g/mol | C6H8O4 | 50 G
Monoethyl fumarate is the monoethyl ester of fumaric acid supplied as a research reagent and reported Nrf2 activator. It is used in biochemical research and as a preservative and polymerization agent for macromolecular materials. The compound is available as a solid and as a 10 mM solution in DMSO for experimental convenience.
- Activates Nrf2 signaling in research assays.
- High reported purity (99.62%).
- Molecular weight 144.13 g/mol and chemical formula C6H8O4.
- Available in multiple pack sizes and solution form.
- Useful as a preservative and polymerization agent for macromolecular materials.
- For research use only; not for clinical use.
Medchemexpress LLC Diroximel fumarate | 1577222-14-0 | ≥98.0% | 255.23 g/mol | C11H13NO6 | 50 MG
Diroximel fumarate is supplied as a research-grade small-molecule reagent intended for laboratory studies. This listing represents a 50 MG pack of the prodrug of monomethyl fumarate and is provided for experimental and analytical use in research settings; it is not for clinical or human use.
- For research use only, not for human or clinical use.
- Supplied as a small 50 MG pack suitable for laboratory testing.
- High purity, typically ≥98.0%.
- Molecular weight 255.23 g/mol and formula C11H13NO6.
- Useful for studies of fumarate metabolism and related biochemical pathways.
Sigma Aldrich Fine Chemicals Biosciences Ketotifen fumarate salt1G
Ketotifen fumarate salt is an antihistamine drug.
