Oxazinanes
![Medchemexpress LLC 4,7-benzothiazoledione, 5-[[2-(dimethylamino)ethyl]amino]-2-methyl- | 477603-18-2 | 99.1% | 10 MG](https://assets.fishersci.com/TFS-Assets/CCG/product-images/5000232564.png-250.jpg)
Medchemexpress LLC 4,7-benzothiazoledione, 5-[[2-(dimethylamino)ethyl]amino]-2-methyl- | 477603-18-2 | 99.1% | 10 MG
BN-82685 (IRC-083065) is a quinone-based CDC25 phosphatase inhibitor used in cell-cycle and cancer research. Supplied as a brown-to-red solid for laboratory research use only.
- Quinone-based CDC25 phosphatase inhibitor used to modulate cell-cycle checkpoints.
- Molecular formula C12H15N3O2S.
- Molecular weight 265.33 g·mol⁻¹.
- CAS number 477603-18-2.
- Appearance: brown to red solid.
- Available in milligram-scale quantities for research applications.
- For research use only; not for human or clinical use.
Medchemexpress LLC iMAC2 hydrochloride | 335166-00-2 | 93.98% | 542.11 | 10 MG
iMAC2 hydrochloride is a potent MAC (mitochondrial apoptosis-induced channel) inhibitor, with an IC50 of 28 nM and a LD50 of 15000 nM. It shows an anti-apoptotic effect and blocks cytochrome c release. It is for research use only and not sold to patients.
- Potent MAC (mitochondrial apoptosis-induced channel) inhibitor
- IC50 of 28 nM
- LD50 of 15000 nM
- Shows anti-apoptotic effect
- Blocks cytochrome c release
Medchemexpress LLC 3-Amino-2-oxazolidinone | 80-65-9 | 98.0% | 102.09 | 10 MG
3-Amino-2-oxazolidinone (AOZ) is a metabolite of Furazolidone used as an indicator for furazolidone residues in vivo. It is orally active and inhibits monoamine oxidase (MAO), increasing monoamine neurotransmitter levels in the brain and lowering blood pressure.
- Used as an indicator for furazolidone residues
- Orally active
- Inhibits monoamine oxidase (MAO)
- Increases levels of monoamine neurotransmitters
- Lowers blood pressure in renal hypertensive rats
Medchemexpress LLC 3-Amino-2-oxazolidinone (AOZ) | 80-65-9 | 98.0% | 102.09 | 10 MG
3-Amino-2-oxazolidinone (AOZ) is a metabolite of Furazolidone. It is used as an indicator for furazolidone residues in vivo and is orally active. In animal models, it has been shown to inhibit monoamine oxidase (MAO) via its metabolite in rat brain and liver, increase monoamine neurotransmitter levels (e.g., norepinephrine and dopamine) in the brain, and lower blood pressure in renal hypertensive rats.
- Used as an indicator for furazolidone residues in vivo.
- Orally active.
- Inhibits monoamine oxidase (MAO).
- Increases monoamine neurotransmitter levels in the brain.
- Lowers blood pressure in renal hypertensive rats.
Medchemexpress LLC 5-Methyl-2-(2H-1,2,3-triazol-2-yl)benzoic acid | 956317-36-5 | 99.99% | C10H9N3O2 | 10 G
5-Methyl-2-(2H-1,2,3-triazol-2-yl)benzoic acid is a chemical compound used as a laboratory reagent and in the manufacture of other substances. This white to off-white solid is characterized by its high purity and specific storage requirements.
- High purity (99.99%)
- Suitable for laboratory chemicals and manufacture of other substances
- Stable as powder at -20°C for 3 years or 4°C for 2 years
- In solvent, stable at -80°C for 6 months or -20°C for 1 month
- Appears as a white to off-white solid
Medchemexpress LLC Clobenpropit dihydrobromide | 145231-35-2 | MFCD00467655 | 99.8% | 470.65 g·mol⁻¹ | C14H19Br2ClN4S | 10 MG
Clobenpropit dihydrobromide is the dihydrobromide salt of clobenpropit, a histamine receptor ligand used for laboratory research. It acts as a potent histamine H3 receptor antagonist/inverse agonist and a partial H4 agonist, with reported additional binding to 5-HT3 and α2 adrenoceptors. The compound is supplied as a high-purity solid for receptor pharmacology and binding studies.
- High purity (99.76%).
- Molecular formula C14H19Br2ClN4S; molecular weight 470.65 g·mol⁻¹.
- CAS number 145231-35-2.
- Potent H3 antagonist/inverse agonist (pEC50 ~8.07).
- Suitable for receptor pharmacology and binding assays.
- Available in small research quantities (e.g., 10 MG).
Medchemexpress LLC (2S,6S)-hydroxynorketamine (hydrochloride) | 1430202-70-2 | MFCD30720898 | 99.3% | 276.16 | C12H15Cl2NO2 | 10 MG
(2S,6S)-Hydroxynorketamine hydrochloride is the hydrochloride salt of the 2S,6S stereoisomer of hydroxynorketamine, a ketamine metabolite widely used as a research reagent in neuropharmacology and mTOR-related studies. Supplied as a white to off-white solid with high reported purity, it is intended for biochemical and cellular assays and is available in milligram-scale pack sizes for laboratory use.
- High reported purity: 99.3%.
- Hydrochloride salt; solid white to off-white appearance.
- Molecular weight 276.16 g/mol.
- Suitable for biochemical and cellular assays in neuropharmacology research.
- Recommended storage: 4°C sealed; in solvent -80°C (6 months) or -20°C (1 month).
- Available in milligram pack sizes, including 10 mg.
Medchemexpress LLC S-2-(4-isothiocyanatobenzyl)-1,4,7,10-tetraazacyclododecane tetraacetic acid | 1020407-41-3 | 99.8% | 551.61 g/mol | C24H33N5O8S | 10 MG
(S)-p-SCN-Bn-DOTA is a bifunctional DOTA-derived chelator used in radiopharmaceutical research. It incorporates an isothiocyanatobenzyl reactive group for covalent attachment to biomolecules and a macrocyclic DOTA core for stable radiometal coordination.
- Enables stable chelation of radiometals for imaging and therapy.
- Provides an isothiocyanate reactive handle for covalent conjugation to proteins and peptides.
- Suitable for labeling studies in small research quantities.
- High chemical purity supports reproducible conjugation and radiolabeling.
- Solid form with recommended cold storage to maintain stability.
TARGETMOL CHEMICALS INC L-778123 HYDROCHLORIDE 25MG
Also available in 2 mg 5 mg 10 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. The L-778123 hydrochloride is an inhibitor of FPTase (IC50 2 nM) and GGPTase-I (IC50 98 nM) in enzyme inhibition determination. purity: 98%
TARGETMOL CHEMICALS INC AFURESERTIB HYDROCHLORID 25MG
Also available in 2 mg 5 mg 10 mg 50 mg 100 mg 200 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Afuresertib hydrochloride is an inhibitor of Akt kinase (Kis of 0.08/2/2.6 nM for Akt1/Akt2/Akt3 respectively)purity: 100%
TARGETMOL CHEMICALS INC SALUBRINAL 25MG
Also available in 2 mg 5 mg 10 mg 50 mg 100 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Salubrinal a phosphatases (PP1) inhibitor(IC50=1.7 uM) exhibits function on the eukaryotic translation initiation factor 2 subunit (eIF2(alpha)). purity: 99%
TARGETMOL CHEMICALS INC JW 55 25MG
Also available in 5 mg 10 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. JW 55 (JW55) is an effective and selective (beta)-catenin signaling pathway inhibitor works by inhibition of the PARP domain of tankyrase 1 and tankyrase 2 (TNKS1/2). purity: 99%
TARGETMOL CHEMICALS INC AZEPEXOLE HYDROCHLORIDE 25MG
Also available in 5 mg 10 mg 50 mg 100 mg 200 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Azepexole hydrochloride (4H-Oxazolo[45-d]azepin-2-amine 6-ethyl-5678-tetrahydro- hydrochloride (11)) is a potent (alpha)2-Adrenoceptor agonist with anaesthetic effects. purity: 99%
TARGETMOL CHEMICALS INC ALVESPIMYCIN HYDROCHLORI 50MG
Also available in 5 mg 10 mg 25 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Alvespimycin hydrochloride (BMS 826476) is a potent HSP90 inhibitor with IC50 of 62 nM. Phase 2. purity: 99%