Cayman Chemical SolIfenacInsuccInate 100mg
A muscarinic M1, M2, and M3 receptor antagonist (Kis = 25, 125, and 10 nM, respectively, for the human receptors); inhibits carbachol-induced calcium mobilization in isolated guinea pig detrusor muscle cells (Ki = 4 nM); inhibits carbachol-induced contraction of isolated guinea pig urinary bladder smooth muscle; inhibits carbachol-induced increases in urinary bladder pressure in anesthetized rats from 0.03-1 mg/kg