Custom Peptides
Cayman Chemical A11trIfluoroacetate salt 10mg
A cell-penetrating peptide; decreases annexin A1 binding to EphA2 and increases EphA2 ubiquitination in HK1 NPC cells; inhibits HK1 and 5-8F NPC cell proliferation, migration, and invasion; reduces tumor volume in 5-8F and HK1 NPC mouse xenograft models
Cayman Chemical 4-acetoxy DMT (hydrochloride), Purity: ≥90%, CAS: 2748484-99-1, 10 mg
An analytical reference standard categorized as a tryptamine; a prodrug form of psilocin; induces the HTR in mice, indicating hallucinogenic potential; intended for research and forensic applications
Cayman Chemical 4-methoxy-α-Pyrrolidinopentiophenone (hydrochloride), Purity: ≥98%, CAS: 5537-19-9, 10 mg
Shares structural features with the stimulant α-PVP, whose mechanism of action is unknown but is believed to act similarly to the designer drug MDPV
Cayman Chemical SB 277011A (hydrochloride), Purity: ≥98%, CAS: 1226917-67-4, 10 mg
A selective antagonist of the dopamine D3 receptor (pKi = 8.0); has high oral bioavailability and enters the central nervous system of the rat
Cayman Chemical 17phenyl trInor ProstglnI 10mg
The 1,15 lactone of 17-phenyl-trinor PGF2α with potential for suitable pharmacologic activity and an improved side-effect profile over current glaucoma therapeutics
Cayman Chemical (+)-Etomoxir (sodium salt), Purity: ≥98%, CAS: 828934-41-4, 10 mg
An inhibitor of CPT1; inhibits fatty acid transport into the mitochondria for β-oxidation; inhibits fatty acid oxidation in hepatocytes in vitro (IC50s = 0.1, 1, and 10 µM for human, guinea pig, and rat hepatocytes, respectively); decreases ATP-linked and uncoupled oxygen consumption in C2C12 myotubes when used in combination with BPTES or UK 5099
Cayman Chemical Phenylpiracetam, Purity: ≥98%, CAS: 77472-70-9, 10 mg
A nootropic derivative of the GABAergic agent piracetam that has been evaluated for its efficacy in reducing neurological deficits related to cerebral ischemia, epilepsy, and neurobehavioral disorders; intended for research and forensic purposes only
Cayman Chemical RCS-4 4-hydroxyphenyl metabolite, Purity: ≥98%, CAS: 1443988-18-8, 10 mg
An expected urinary metabolite of RCS-4 that is potentially useful as a metabolic marker for the identification of RCS-4 ingestion; intended for research and forensic purposes
Cayman Chemical 2-Phenethylamine (hydrochloride), Purity: ≥98%, CAS: 156-28-5, 10 mg
A natural monoamine alkaloid that acts as neuromodulator in the central nervous system; stimulates the release of norepinephrine and dopamine and is metabolized by monoamine oxidases as well as other enzymes; intended for forensic and research applications
Cayman Chemical Khasianine, Purity: ≥98%, CAS: 32449-98-2, 10 mg
A steroidal glycoside with diverse biological activities; reduces the proliferation of LNCaP and T47D cancer cells (IC50s = 32.1 and 27.5 µM, respectively); inhibits TNF-α-induced nuclear translocation of NF-κB in HaCaT keratinocytes at 50 nM; decreases AST serum levels in a mouse model of carbon tetrachloride-induced liver injury at 0.1 mg/kg; topical administration reduces ear epidermal thickness and scaling, as well as leukocyte and macrophage infiltration, in an imiquimod-induced mouse model of psoriasis at 5 mg/kg
Cayman Chemical Moexiprilat, Purity: ≥95%, CAS: 103775-14-0, 10 mg
An ACE inhibitor and active metabolite of the prodrug moexipril (IC50 = 2.1 nM); prevents the estrone- or angiotensin II-stimulated proliferation of primary neonatal rat cardiac fibroblasts at 10 nM; reduces mean arterial blood pressure and increases the levels of atrial natriuretic peptide in ovariectomized mice at 50 mg/kg per day
Cayman Chemical N8-Acetylspermidine (hydrochloride), Purity: ≥95%, CAS: 34450-15-2, 10 mg
An endogenous polyamine; urinary levels are increased in patients with chronic pancreatitis; blood levels are increased in patients with ischemic cardiomyopathy, as well as in patients with Parkinson’s disease
Cayman Chemical S1HtrIfluoroacetate salt 10mg
A synthetic peptide antagonist of the human growth hormone receptor; decreases STAT5 phosphorylation induced by human growth hormone in SK-MEL-28 and MALME-3M cell lines, as well as by prolactin in IM-9 B cells, at 100 and 200 nM
Cayman Chemical CaMKII-IN-1, Purity: ≥95%, CAS: 1208123-85-6, 10 mg
A CaMKII inhibitor (IC50 = 0.063 µM); is selective for CaMKII over CaMKIV, MLCK, p38α, Akt1, and PKC (IC500s = >60, 36, 11, 30, and 21 µM, respectively)
Cayman Chemical Florfenicol amine (hydrochloride), Purity: ≥95%, CAS: 108656-33-3, 10 mg
A metabolite of florfenicol